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2-methoxy-N-({5-[(2,4,6-trifluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[3-(pyridin-3-yloxy)propyl]acetamide
N-{2-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}acetamide
3-(2-methylpropyl)-N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-1,2-oxazole-5-carboxamide
1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(pyridin-3-ylmethyl)piperazine
4-hydroxy-N-{[3-(methylcarbamoyl)-1,2,4-oxadiazol-5-yl]methyl}-2-phenylpyrimidine-5-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
2-fluoro-4-methyl-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)benzamide
1-(pyridin-3-ylmethyl)-4-[4-(trifluoromethyl)benzoyl]-1,4-diazepane
3-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-chlorophenyl)urea
3-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline
N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-oxo-1-(2-phenylethyl)-N-(propan-2-yl)piperidine-3-carboxamide
N-[2-(3-methoxyphenyl)ethyl]-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
4-fluoro-N-(2-{7-[(2E)-2-methylbut-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
5-(3,4-dimethylphenoxymethyl)-N-[2-(2-oxopiperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
1-(butan-2-yl)-N3-butyl-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(3aR,6aR)-2-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-phenyl-1-[3-(phenylamino)piperidin-1-yl]butane-1,2-dione
1-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-3-(1H-1,2,4-triazol-3-yl)urea
2-(3-methoxypropyl)-8-[3-(pyridin-4-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
1-methyl-2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1H-imidazole
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-ethyl-1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidine-3-carboxamide
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-[(5-methylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2,5-dioxo-6-[4-(pyridin-2-yl)butyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-({methyl[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amino}methyl)-N-(6-methylpyridazin-3-yl)benzamide
dimethyl[(1-{1-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]amine
[(6-methylpyridin-2-yl)methyl]({[2-(morpholin-4-yl)pyridin-3-yl]methyl})amine
1-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(4-ethylpiperazin-1-yl)ethan-1-one
5-[(2-chlorophenyl)methyl]-5-[1-(2-cyclopentylacetyl)piperidin-4-yl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
2-[3-(2-chlorophenyl)-1,2-oxazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
dimethyl(2-{2-[1-(morpholine-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-phenyl-1,2,4-oxadiazole
ethyl 1-[(2-hydroxyphenyl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(2-methylprop-2-en-1-yl)acetamide
2,7-dioxo-N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-1,3-diazepane-4-carboxamide
2-(2,3-difluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
(3R,4R)-4-methyl-1-(5-phenyl-1,2,4-oxadiazol-3-yl)-3-(propan-2-yl)pyrrolidin-3-ol
6-methyl-3-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-methyl-8-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
4-(3-{7-[ethoxy(phenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl}phenyl)-2-methylbut-3-yn-2-ol
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-(1-methyl-1H-pyrazol-4-yl)propanamide
5-chloro-2-{3-[2-(furan-3-yl)-1H-imidazol-1-yl]propyl}-1H-1,3-benzodiazole
N-(2-methoxyethyl)-1-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
5-methoxy-3-{[4-(piperidine-1-carbonyl)piperidin-1-yl]methyl}-1H-indazole
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
1-[(diethylcarbamoyl)methyl]-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidine
ethyl 4-[(4-methoxyphenyl)methyl]-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxylate
3-[(4aR,7aS)-4-[2-(azepan-1-yl)-2-oxoethyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid