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N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
diethyl({2-ethyl-5-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]furan-3-yl}methyl)amine
2-methyl-5-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
1-ethyl-N-methyl-5-[(3-methylbutyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2S,4R)-4-[(4-methoxyphenyl)sulfanyl]-1-[(2-methyl-1H-indol-3-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidine-3-carboxamide
N-(1,4-dioxan-2-ylmethyl)-2-(trifluoromethyl)benzamide
[(3-{2-[4-(2,2-dimethyloxane-4-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](1H-imidazol-2-ylmethyl)methylamine
N-(oxolan-2-ylmethyl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-propylbenzamide
1-(2-methylpropyl)-5-(thiophen-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
(3E)-N-{[1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrrolidin-3-yl]methyl}pent-3-enamide
N-({1-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]pyrrolidin-3-yl}methyl)methanesulfonamide
N-[1-(4-fluorophenyl)propyl]-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanamide
2-amino-6-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-(2-methoxypyrimidin-5-yl)pyridine-3-carbonitrile
N-[1-(3,5-difluorophenyl)ethyl]-4-hydroxy-1-methylpiperidine-4-carboxamide
4-(1-methyl-1H-imidazol-5-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}pyrimidine-5-carboxylic acid
2-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
1-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-2-(2,3-dimethylphenoxy)ethan-1-one
2-benzyl-5-formamido-1-methyl-N-[2-(pyridin-3-yloxy)propyl]-1H-1,3-benzodiazole-7-carboxamide
2-[(4-chlorophenyl)methyl]-8-(3-methyl-1,2-oxazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-[(1,4-dithiepan-6-yl)amino]-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
1-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(4-chloro-1H-pyrazol-1-yl)ethan-1-one
9-(oxolan-3-ylmethyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3S)-N,N-dimethyl-1-(quinoxalin-2-yl)azepan-3-amine
1,4-dimethyl-9-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-1,4,9-triazaspiro[5.5]undecane
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
2-(1H-imidazol-1-yl)-1-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-(4-methoxyphenyl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}cyclopentane-1-carboxamide
1-tert-butyl-N-(2-hydroxyethyl)-5-oxo-N-(1,3-thiazol-2-ylmethyl)pyrrolidine-3-carboxamide
N-ethyl-2-hydroxy-5-methoxy-N-[2-(3-methoxyphenoxy)ethyl]benzamide
(2S)-1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}pyrrolidine-2-carboxamide
N-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxan-4-amine
3-methyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-1H-pyrazole-5-carboxamide
N-({1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]piperidin-4-yl}methyl)acetamide
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
1-{2-[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[4-(benzenesulfonyl)phenyl]-1H-pyrrolo[2,3-b]pyridine
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(1-methyl-1H-pyrazol-4-yl)propanamide
N-[1-(4-methanesulfonylphenyl)propyl]-2,3-dihydro-1H-inden-2-amine
4-{1-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}thiomorpholine
7-methyl-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
2-{4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
5-methyl-1'-[3-(1H-pyrazol-1-yl)benzoyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{4-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]phenyl}acetic acid
[4-(azepan-1-yl)butyl][2-methyl-2-(morpholin-4-ylmethyl)propyl]amine
(1S,5R)-6-(2-methoxyethyl)-3-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-ethyl-2-[1-(3-methylbutyl)-1H-pyrazol-4-yl]benzamide
3-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
(3S,5S,9R)-5-{[(3-chloro-1-benzothiophen-2-yl)methyl]amino}-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione