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2-{3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl}pyrazine
2-(2-methyl-1H-1,3-benzodiazol-1-yl)-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
5-ethyl-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-1,3-oxazole-4-carboxamide
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]propanamide
{3-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-3-oxopropyl}urea
(2S,4S)-1-methyl-4-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}pyrrolidine-2-carboxylic acid
1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
4-(2,5-dimethoxyphenyl)-5-methylthieno[2,3-d]pyrimidine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-(1H-indol-5-ylmethyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-[(2-chlorophenyl)methyl]-N-[3-(methylsulfanyl)propyl]-1H-1,2,3-triazole-4-carboxamide
1-cyclopentyl-4-[4-(morpholin-4-yl)benzoyl]-1,4-diazepane
3-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-1,4-oxazepan-6-yl)methanol
N-[3-(1,3-benzothiazol-2-yl)propyl]-1H-pyrazole-4-carboxamide
N-[2-(2-ethoxyphenoxy)ethyl]-N-methyl-2-(1H-1,2,4-triazol-1-yl)propanamide
7-(2-methylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
(1S,5R)-6-(2-ethylpyridine-4-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
3-(1-methyl-1H-1,2,3-triazol-4-yl)-1-[1-(thian-4-yl)piperidin-4-yl]urea
2-(dimethyl-1,2-oxazol-4-yl)-1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}ethan-1-one
2-[3-(methoxymethyl)phenyl]-2-{4-[(2-methylphenyl)methyl]piperazin-1-yl}acetic acid
2-{[(1S,3aS,6aS)-octahydropentalen-1-yl]amino}pyridine-3-carboxylic acid
N5-methyl-N5-(oxan-4-ylmethyl)-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N,N-bis(prop-2-en-1-yl)-2-[(prop-2-yn-1-yl)amino]acetamide
1-benzyl-4-(2,6-dimethoxypyridine-3-carbonyl)-1,4-diazepan-6-ol
2-{6-chloro-2-methylimidazo[1,2-a]pyridine-3-carbonyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-acetyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)thiophene-3-carboxamide
1-(2-chlorophenyl)-4-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)piperazin-2-one
N-(3-methyl-1-{7-[(5-methylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}pyridine-2-carboxamide
6-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-N,N-dimethylpyridine-3-carboxamide
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-(3-methoxyphenyl)pyrrolidine
6-amino-N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]pyridine-3-carboxamide
8-chloro-2-{[methyl({[2-(methylamino)pyrimidin-5-yl]methyl})amino]methyl}quinolin-4-ol
1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-(4-fluorophenyl)piperidin-3-amine
N-({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)-N-(prop-2-yn-1-yl)cyclohexanamine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-1H-indole-6-carboxamide
N-[(3R,4R)-1-(1,3-benzothiazol-2-yl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-4-(trifluoromethyl)pyrimidin-2-amine
1-methyl-6-(pyridin-4-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-(4-methoxyphenyl)-N-methyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
7-[(4-methanesulfonylphenyl)methyl]-2,7-diazaspiro[4.5]decane
4-hydroxy-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
4-({[2-(azepan-1-yl)ethyl](methyl)amino}methyl)-5-(hydroxymethyl)-2-methylpyridin-3-ol
4-{4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-1-yl}-1-propylpiperidine
1-(cyclohexylmethyl)-3-(oxan-4-yl)-5-(pyrrolidin-3-yl)-1H-1,2,4-triazole
N-[(1R)-2,3-dihydro-1H-inden-1-yl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N,1-dimethyl-6-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,6-dihydropyridazine-3-carboxamide
2,6-dimethyl-N-(morpholin-2-ylmethyl)pyridine-4-carboxamide