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1-[(4-ethylphenyl)methyl]-4-[2-(thiomorpholine-4-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
3-chloro-N-(2-methoxyethyl)-4-{[1-(prop-2-en-1-yl)piperidin-4-yl]oxy}benzamide
(1R,6S)-9-methyl-3-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-3,9-diazabicyclo[4.2.1]nonane
1-{4-[(5-hydroxy-4,4-dimethylpentyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
(3S,4S)-1-[(4-phenylphenyl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-{1-[1-(oxolane-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
1-{2-oxo-2-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethyl}azepan-2-one
2-methyl-9-(4-methylpiperazine-1-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2-cyclopentylacetyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-{[1-(oxan-4-yl)pyrrolidin-3-yl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
1-(cyclopropylmethyl)-4-(2,3-dihydro-1-benzofuran-7-carbonyl)-2-(propan-2-yl)-1,4-diazepane
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
7-[2-(ethylamino)pyrimidine-5-carbonyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 5-cyano-6-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-methylpyridine-3-carboxylate
1-(2-chloroprop-2-en-1-yl)-7-fluoro-3-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
3-[(4-methyl-1,3-thiazol-5-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
2-[({2-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)amino]propane-1,3-diol
2-({[(3R,4R)-1-[5-chloro-3-(trifluoromethyl)pyridin-2-yl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}pyridine-3-carboxylic acid
2-(cyclopropylmethyl)-8-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-cyclopropyl-N-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-amine
2-[4-({2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)-3-methyl-1H-pyrazol-1-yl]ethan-1-ol
1-methyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-(morpholin-4-yl)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-oxopentanamide
3-phenyl-4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,2-oxazole
1-(4,7-dimethylquinazolin-2-yl)-N-[(2-methylphenyl)methyl]piperidine-4-carboxamide
1-methyl-5-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-1H-indole
2-{4-[(2-methylphenyl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-(2,2-dimethylpropanoyl)-4'-(3-methylbutyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-cyclopropyl-N-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}-4-methylbenzamide
methyl 6-[4-(2-methoxyphenoxy)piperidin-1-yl]pyrimidine-4-carboxylate
3-(5-chloro-2-methoxypyridin-4-yl)-N-methylpyrazin-2-amine
6-(2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)-2-methylpyrimidin-4-ol
1-(2-phenylethyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
3-({[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]amino}methyl)pyrrolidin-3-ol
4-[4-({7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecan-3-yl}methyl)phenyl]-2-methylbutan-2-ol
1-[(3-methyl-1-benzofuran-2-yl)methyl]-4-(thian-4-yl)piperazine
1-[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]-2,2-diphenylethan-1-one
3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}propanamide
(3S,4R)-4-(2-methylphenyl)-1-(quinoline-3-carbonyl)pyrrolidine-3-carboxylic acid
2-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-6-methoxyphenoxy)propanoic acid
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-(pyridin-3-yl)acetamide
2-amino-4-ethyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1,3-thiazole-5-carboxamide
N-methyl-3-phenyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-oxazole-4-carboxamide
2-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}furan-2-carboxamide
4-(4-fluorophenyl)-4-hydroxy-N-(2-methoxy-6-methylphenyl)piperidine-1-carboxamide
1-(2-methyl-1-benzofuran-5-carbonyl)-3-(1-methyl-1H-imidazol-2-yl)piperidine