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2-cyclohexyl-6-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,3-benzoxazole
N-{1-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
methyl 3-(1H-pyrazol-3-yl)benzoate
2-[(furan-3-ylmethyl)(pyridin-2-ylmethyl)amino]-2-methylpropan-1-ol
ethyl 1-(2-methylpropyl)-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-({[(3R,4R)-1-[(2-fluoro-4-methylphenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(1S,5R)-6-(cyclobutylmethyl)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamide
3-ethyl-1-[4-(hydroxymethyl)cyclohexanecarbonyl]piperidine-3-carboxylic acid
1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-4-(pyridin-3-ylmethyl)piperazine
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[2-(5-methylthiophen-2-yl)ethyl]benzamide
5-[1-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,3,4-thiadiazol-2-amine
2-methyl-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1,3-benzothiazole-6-carboxamide
2-({1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}methyl)-1H-1,3-benzodiazole
3-{[(2,3-dihydroxypropyl)amino]methyl}-1-[(4-methoxyphenyl)methyl]-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
methyl (2S,4S)-4-(furan-2-amido)-1-[(2-methylphenyl)methyl]pyrrolidine-2-carboxylate
3-methoxy-N-{1-[7-(quinolin-7-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
(2,3-dihydro-1-benzofuran-2-ylmethyl)({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})methylamine
1-methyl-9-(prop-2-en-1-yl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[(2,3-difluoro-4-methylphenyl)methyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
(3S)-4-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
4-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}-2,6-dimethoxyphenol
1-(2-{1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]pent-4-enamide
N-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-azabicyclo[2.2.2]octan-3-amine
[(5-ethylpyridin-2-yl)methyl][(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amine
ethyl 4-{6-[4-(1H-pyrazol-1-yl)benzoyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
[(3R,4R)-1-(2,4-dimethoxybenzoyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
1-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-methylbut-2-en-1-one
3-[(3-chlorophenyl)methyl]-N-(1,4-dioxan-2-ylmethyl)-N-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-(1H-pyrazol-4-yl)butanamide
6-(2,5-dimethylfuran-3-yl)-N-(2-methoxyethyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-cyclopropyl-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-hydroxypyrimidine-5-carboxamide
(3R,4S)-4-[ethyl({2-methylthieno[2,3-d]pyrimidin-4-yl})amino]oxolan-3-ol
2-(2-aminopyrimidin-5-yl)-N,N,3,6-tetramethylquinoline-4-carboxamide
3-(oxolan-3-yl)-5-(5-phenyl-1,2-oxazol-3-yl)-1,2,4-oxadiazole
4-(2-chloro-4-fluorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
1-methyl-N-[(1R,3S)-3-{[3-(methylsulfanyl)phenyl]carbamoyl}cyclopentyl]-1H-pyrrole-2-carboxamide
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-(thiophen-3-ylmethyl)pyrimidine-5-carboxamide
1-(4-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
2-(3-methoxyphenyl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1,3-benzoxazole-6-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one
5,6-dimethoxy-2-[(2-methyl-1,3-oxazol-4-yl)methyl]-1,2-dihydroisoquinolin-1-one
(1R,4S)-2-[2-(pyridin-4-yl)pyridine-3-carbonyl]-2-azabicyclo[2.2.1]heptane
(1S,5R)-3-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopropyl-5-(dimethoxy-1,3,5-triazin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-(3-amino-6-methoxy-1H-indazol-1-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
4-methanesulfonyl-2-(4-methylpentyl)morpholine