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6-[3-(cyclopropylmethyl)-1-ethyl-1H-1,2,4-triazol-5-yl]quinoxaline
2-hydroxy-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-4-(methylsulfanyl)butanamide
2-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
4-(cyclopropylmethyl)-1-[(5-ethylpyridin-2-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
4-[(2,4-difluorophenyl)methyl]-9-methoxy-7-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(piperidine-4-carbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-3-yl)ethan-1-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-fluoro-2-[2-(1H-imidazol-1-ylmethyl)pyrrolidin-1-yl]pyrimidin-4-ol
4-{1-[2-(furan-3-yl)-1H-imidazol-1-yl]butan-2-yl}morpholine
1-{[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}piperidine-3-carbonitrile
N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-2,1-benzoxazole-3-carboxamide
(2R,3S,6R)-3-phenyl-5-[3-(pyridin-3-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
(3aR,5R,6S,7aS)-2-{[5-(2-chlorophenyl)furan-2-yl]methyl}-octahydro-1H-isoindole-5,6-diol
8-(3-chloro-4-hydroxybenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N,N-dimethyl-5-[1-(propan-2-yl)piperidine-3-carbonyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
[2-(1H-1,3-benzodiazol-2-yl)ethyl](ethyl)[(1-ethyl-1H-pyrazol-4-yl)methyl]amine
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-ethylbutan-1-one
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-(2-methylpropyl)-5-(6-methylquinolin-5-yl)furan-2-carboxamide
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(furan-2-ylmethyl)(prop-2-yn-1-yl)amine
2-{1-[(2-ethoxyphenyl)methyl]-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
3-[5-(3-chlorobenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-(propan-2-yl)propanamide
N-[2-(furan-2-yl)ethyl]-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
dimethyl(2-{[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl](thiophen-3-ylmethyl)amino}ethyl)amine
N-(2,4-dimethoxyphenyl)-3-(4-methoxy-2-methylbenzoyl)piperidine-1-carboxamide
ethyl 3-({1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)propanoate
2-methoxy-N-(1-{1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
3-methyl-1-(2-methylpropyl)-8-[3-(methylsulfanyl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-[(3,4-difluorophenyl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
4-(2-methoxyethyl)-11-{[(4-phenyloxan-4-yl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-benzyl-N-ethyl-2-[3-(3-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]acetamide
N-[2-(4-ethylmorpholin-2-yl)ethyl]-3,5-dimethyl-1H-indole-2-carboxamide
6-(aminomethyl)-2-(4-chlorophenyl)-3,4-dihydropyrimidin-4-one
1-ethyl-N-methyl-5-[(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(azepan-1-yl)-3-(4-chloro-2-{[(prop-2-en-1-yl)amino]methyl}phenoxy)propan-2-ol
2-{3-[4-(3-chlorophenyl)piperazin-1-yl]propyl}-5-(dimethylamino)-2,3-dihydropyridazin-3-one
(4aS,7aR)-1-(3,5-dimethoxybenzoyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-chloro-2-(4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
(3S,5R,9R)-11-[(2-fluoro-5-methylphenyl)methyl]-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N-[(3S,4R)-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
N-[(3S)-2-oxoazepan-3-yl]-2-(2-phenyl-1,3-thiazol-4-yl)-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}acetamide
N-ethyl-N-methyl-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
N-(2-ethylbutyl)-1-(morpholin-4-ylmethyl)cyclohexan-1-amine
(2R,3R,6R)-3-phenyl-5-(quinoline-8-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-({1-[2-amino-6-(propan-2-yl)pyrimidine-4-carbonyl]piperidin-3-yl}methyl)-4-fluorobenzamide
4-[6-(piperidin-1-yl)pyrimidin-4-yl]-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-[2-(2,4-difluorophenyl)ethyl]-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidine
3-methyl-8-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one