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N-methyl-N-[(1-methylpiperidin-3-yl)methyl]-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
(3aS,6aR)-5-(2H-1,3-benzodioxol-4-ylmethyl)-3-[2-(4-fluorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(3S,4S)-1-[(2-ethoxynaphthalen-1-yl)methyl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
2-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-2-(morpholin-3-yl)acetamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]pyrrolidin-3-yl]methanol
2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]acetamide
N-(1-{7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
4-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(1-methylpiperidin-3-yl)methyl]furan-2-carboxamide
(1R,5S,6R)-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-{3-[(4-methylphenyl)sulfanyl]propyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-(1-{4-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)oxane-4-carboxamide
2-[2-(3-benzyl-1H-1,2,4-triazol-5-yl)ethyl]-1-methylpiperidine
4-[4-(furan-2-yl)benzoyl]-7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(2,4-difluorophenyl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-phenoxy-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]benzamide
N-(4-{1-[2-(methylsulfamoyl)ethyl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide
N-methyl-N-{2-phenyl-1-[1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]ethyl}pyridine-2-carboxamide
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}oxolane-3-carboxamide
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-1,4-diazepane
2-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}pyridin-3-ol
1,3-dimethyl-5-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-N,N-dimethylpiperidin-3-amine
[3-(3-phenylpropyl)-1-(quinolin-2-ylmethyl)piperidin-3-yl]methanol
2-{4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-(5-methyl-1,3-oxazole-4-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
3-(4-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)-1H-pyrazol-5-ol
3-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-1-(3-sulfamoylphenyl)urea
1-ethyl-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-{2-[2-(4-fluorophenyl)azetidin-1-yl]-2-oxoethyl}-3-methyl-1,2-dihydroquinoxalin-2-one
3-(4-chlorophenyl)-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
{4-benzyl-1-[4-(4-methoxyphenyl)butan-2-yl]piperidin-4-yl}methanol
1-[(2-ethylpyrimidin-5-yl)methyl]-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
5-{[4-(2-methylphenyl)-1,4-diazepan-1-yl]methyl}quinoxaline
2-(4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)-1-(pyrrolidin-1-yl)ethan-1-one
2-methoxy-N-[1-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
ethyl 4-[(4-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperazine-1-carboxylate
N-{2-[(4-methoxyphenyl)sulfanyl]ethyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
3-ethoxy-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
N-[(4-hydroxy-6-methylpyrimidin-2-yl)methyl]-4-(methylsulfanyl)benzamide
1-methyl-N-[1-(morpholin-4-ylmethyl)cyclopentyl]-3-propyl-1H-pyrazole-5-carboxamide
5-(1-butyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
6-{[2-(3-phenylpropyl)morpholin-4-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N,2-diethyl-N-methyl-7-{[(1s,4s)-4-aminocyclohexyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(5-ethylpyridin-2-yl)methyl]-N,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[1-(1H-indole-6-carbonyl)piperidin-3-yl]benzoic acid
N-(4-fluorophenyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-amine
ethyl 4-[6-(1H-indol-2-ylmethyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
3-({2-methyl-3-[(pyridin-2-ylmethyl)amino]phenyl}formamido)butanoic acid