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2-amino-4-ethyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1,3-thiazole-5-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[(4-methylphenyl)methyl]-1H-pyrazole-4-carboxamide
(4aR,8aR)-7-[(3-chlorophenyl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
1-cyclohexyl-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]piperidine-4-carboxamide
2-(7-methoxy-4-methylquinazolin-2-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
4-({1-[2-(1H-1,2,4-triazol-1-yl)acetyl]pyrrolidin-3-yl}methyl)benzoic acid
1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-methoxyethyl)methylamine
1-[(3-fluoro-4-methylphenyl)methyl]-5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
1-(3-cyano-4-methylphenyl)-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
4-(6-methylpyridin-2-yl)-N-[3-(methylsulfamoyl)phenyl]piperazine-1-carboxamide
1-(4,6-dimethylpyrimidin-2-yl)-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-phenyl-1,4-diazepane
(3aS,6aS)-2-cyclopentyl-5-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(1-benzothiophen-2-ylmethyl)-N-methyl-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidine-2-carboxamide
2-(2-phenoxyethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-{[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]oxy}-N-[2-(dimethylamino)ethyl]-N-methylbenzamide
3-{1-[1-(methoxymethyl)cyclopropanecarbonyl]piperidin-3-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}isoquinoline
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methylpyrazin-2-yl)methyl]acetamide
6-[4-(2-methoxyethoxy)phenyl]-3,4-dihydroquinazolin-4-one
1-(5-ethyl-1,2-oxazole-3-carbonyl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
6-(2,6-dimethylquinoline-4-carbonyl)-N-[3-(1H-imidazol-1-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
N,N-dimethyl-3-[4-(pyridin-3-yl)piperazine-1-carbonyl]piperidine-1-carboxamide
5-(methoxymethyl)-N-{[5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
4,6-dimethyl-2-oxo-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,2-dihydropyridine-3-carboxamide
5-[({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]pyrimidin-2-amine
3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methyl-4-phenylpyridine
3-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-oxazolidin-2-one
4-({3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}methyl)quinoline
4-(4-benzyl-1H-1,2,3-triazol-1-yl)-1-(1,2-oxazole-3-carbonyl)piperidine
2-methyl-3-(2-{4-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}ethyl)quinolin-4-ol
2-(1-methyl-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl)ethan-1-ol
(4aR,8aS)-1-[2-(dimethylamino)ethyl]-6-(3-phenylpropyl)-decahydro-1,6-naphthyridin-2-one
2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-5-methylpyrazine
3,6-dimethyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
5-acetyl-N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}thiophene-2-carboxamide
N-methyl-N-[(5-methylfuran-2-yl)methyl]-1H-indole-3-carboxamide
2-[(4-chlorophenyl)methyl]-8-(oxolan-3-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
2-(4-methanesulfonylphenyl)-1-[4-(1H-pyrazol-5-yl)phenyl]-1H-imidazole
1-(3-carbamoylpyridin-2-yl)-4-[(4-chlorophenyl)methyl]piperidine-4-carboxylic acid
1-ethyl-8-(1-hydroxypropan-2-yl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cycloheptyl-N-[(1-hydroxycyclohexyl)methyl]-6-oxopiperidine-3-carboxamide
1-{4-[4-(1-hydroxycyclopentyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-3-(1-methylcyclopropyl)propan-1-one
5-(piperidin-4-yl)-3-[2-(propan-2-ylsulfanyl)ethyl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
[4-fluoro-3-(2-fluoro-3-methoxyphenyl)phenyl]methanamine
1-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-2-(dimethyl-1H-1,2,4-triazol-1-yl)ethan-1-one
N-({5-[(oxolan-2-ylmethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)cyclohexanecarboxamide
2-(dimethylamino)-N-[2-(4-fluorophenyl)-1-[1-(1-methyl-1H-indole-2-carbonyl)piperidin-4-yl]ethyl]-N-methylacetamide
10-methoxy-5-(5-phenyl-1,2-oxazole-3-carbonyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine