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3-[(3-methyloxetan-3-yl)methyl]-1-(2,3,5-trifluorophenyl)urea
1-(4-{[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}thiophen-2-yl)ethan-1-one
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-N-(pyridin-3-ylmethyl)oxolane-2-carboxamide
ethyl 5-[1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(4-{[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
3-oxo-N-[1-(pyridin-2-yl)propan-2-yl]-2,3-dihydro-1H-indene-1-carboxamide
2-(4-chlorophenyl)-1-[2-(oxan-2-yl)ethyl]-1H-imidazole
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1S,5R)-6-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(1R,2R,6S,7S)-4-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-azatricyclo[5.2.1.02,6]decane
1-[(5-chlorofuran-2-yl)methyl]-2-(pyrrolidin-1-ylmethyl)piperidine
1-(cyclopropylmethyl)-N-(pyridin-2-ylmethyl)-5-(2,2,3,3-tetramethylcyclopropanecarbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-2-(pyridin-4-ylsulfanyl)acetamide
1-[(1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
4-[3-(morpholin-4-ylmethyl)piperidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
ethyl 4-oxo-5-phenoxy-1-[(1R,2S)-2-phenylcyclopropyl]-1,4-dihydropyridine-3-carboxylate
N-[(1-acetylpiperidin-3-yl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-ethyl-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]propanamide
1-[3-(methylsulfanyl)propanoyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
5-[(4-cyclohexyl-3-oxopiperazin-1-yl)methyl]-2-methoxybenzoic acid
N3-[3-(4-ethoxyphenyl)propyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
(4aR,7aS)-1-[(5-methylfuran-2-yl)methyl]-4-(1,2-oxazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
9-[(3E)-pent-3-enoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine
1-[(2-fluorophenyl)methyl]-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
(2,2-dimethyl-3-{2-[2-(morpholin-4-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}propyl)dimethylamine
2-(2-{1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1H-imidazol-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(2-methylphenyl)-3-{2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl}-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
2-(3-{[3-(2-phenylacetyl)piperidin-1-yl]methyl}phenoxy)acetamide
3-amino-1-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-(naphthalene-1-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
5-{9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carbonyl}pyridine-2-carbonitrile
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]oxolane-3-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{3-[(5-methylpyridin-2-yl)amino]propyl}acetamide
methyl 2-(phenylsulfamoyl)-6-[(3,4,5-trifluorophenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-methyl-N-(pyridin-3-ylmethyl)-4-{[1-(thiophen-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-cyclopropyl-N-[1-(phenylcarbamoyl)piperidin-4-yl]pyrimidine-5-carboxamide
1-benzyl-6-(cyclopropylmethoxy)-4-(5-hydroxy-4-oxo-4H-pyran-2-carbonyl)-1,4-diazepan-2-one
2-(4-{[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]methyl}phenoxy)propanoic acid
1-[(3S,4R)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
2-methoxy-1-[1'-(3-methyl-1,2-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-(furan-2-ylmethyl)-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-2,3-dihydro-1H-indol-2-one
5-acetyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]thiophene-3-carboxamide
2-cyclopropyl-8-[(1-methyl-1H-indol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazin-1-yl)pyrazine
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
2-[4-(5-chloro-2-methylpyrimidine-4-carbonyl)piperazin-1-yl]-1,3-benzothiazole