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2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
7-chloro-2-{[methyl(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amino]methyl}-N-(oxolan-2-ylmethyl)quinazolin-4-amine
1-[1-(2-phenylethyl)-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
3-(2-chlorophenyl)-N-methyl-N-(oxan-4-yl)-3-phenylpropanamide
1,3,7-trimethyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-1H-indole-2-carboxamide
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-ethyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2,3-dihydro-1-benzothiophene-2-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-cyclohexylpyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]isoquinoline
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-{4-[2-(dimethyl-1,3-thiazol-4-yl)acetamido]-2-methoxyphenyl}butanamide
2-(4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperazin-1-yl)-1,3-benzoxazole
N-benzyl-2,4-dimethyl-N-(1,3-thiazol-2-ylmethyl)pyrimidine-5-carboxamide
2-{5-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazol-5-yl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-ethyl-N-(furan-3-ylmethyl)-N,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-({[(4-fluorophenyl)methyl](1-methoxypropan-2-yl)carbamoyl}amino)-N-methylbenzamide
3-{1-[(6-chloroquinolin-2-yl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
(3S,4S)-1-[2-(cycloheptylcarbamoyl)ethyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]acetamide
1-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-3-methyl-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(furan-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(4-phenylpiperidin-1-yl)acetamide
N4-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}pyrimidine-4,6-diamine
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,2,7,8-tetramethylquinoline-4-carboxamide
2-methyl-1-(5-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophen-2-yl)propan-1-one
2-{1-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-4-yl}-5-fluoro-1H-1,3-benzodiazole
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
3-(1-ethyl-1H-pyrazol-3-yl)-4-(3-methylphenyl)-4H-1,2,4-triazole
4-cyclobutyl-2-[(3-methoxyphenyl)methyl]morpholine
N-[(4-chlorophenyl)methyl]-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
2-(azepan-1-yl)-N-[2-(1H-imidazol-4-yl)ethyl]acetamide
3-(morpholine-4-carbonyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]benzene-1-sulfonamide
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]acetamide
1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-3-(thiophene-2-carbonyl)piperidine
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
2-{9-[(3-cyanophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
1-butyl-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-1-[(5-methylthiophen-2-yl)methyl]urea
methyl 5-[(5-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-{1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]pyrrolidin-2-yl}-1,3-benzothiazole
(3R,4R)-4-amino-1-{3-[(3-fluorophenyl)methoxy]benzoyl}piperidin-3-ol
(1S,5R)-1,3,3-trimethyl-N-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}-6-azabicyclo[3.2.1]octane-6-carboxamide
3-hydroxy-N-[3-(phenylsulfanyl)propyl]benzamide
6-fluoro-3-[1-(1H-pyrazol-1-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
1-(1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}piperidin-3-yl)-2-phenylethan-1-one
5-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
2-(2-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}phenoxy)acetic acid
N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
3-({[(4-chlorophenyl)methyl]amino}methyl)-3-hydroxy-1-(2-phenylethyl)piperidin-2-one