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N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
N-(2-methoxyethyl)-1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperazine-2-carbonyl}morpholine
ethyl 1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4-(2-phenylethyl)piperidine-4-carboxylate
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-(3-fluoro-4-methoxybenzoyl)-7-azaspiro[3.5]nonan-1-ol
4-methyl-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
7-{[4-(methylsulfanyl)phenyl]methyl}-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
1-[3-(pyridin-4-yl)azetidin-1-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)ethan-1-one
3-(but-2-yn-1-yl)-5-(2-phenylethyl)-5-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
N'-(5-methyl-1,2-oxazol-3-yl)-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]ethanediamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
3-(4-fluorophenyl)-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazin-2-one
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
ethyl 4-[(2-chlorophenyl)methyl]-1-(pyridine-4-carbonyl)piperidine-4-carboxylate
3-(pyrrolidin-1-ylmethyl)-1-(quinoline-4-carbonyl)piperidin-3-ol
methyl[(3-methylthiophen-2-yl)methyl]{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
2-(4-methoxyphenyl)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
ethyl 3-[({1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}carbamoyl)amino]propanoate
N-ethyl-2-(4-{5-[(4-methylpiperidin-1-yl)methyl]furan-2-carbonyl}piperazin-1-yl)acetamide
1-(1-cyclopentyl-6-oxopiperidine-3-carbonyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(oxolane-2-carbonyl)piperidine-4-carboxylic acid
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-6-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[3-({[(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amino}methyl)phenoxy]acetamide
4-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-2-ethylpyrimidine
1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-(2-phenylethyl)piperidine
(1R,3S)-3-methoxy-7-(2,4,5-trimethoxybenzoyl)-7-azaspiro[3.5]nonan-1-ol
N-[(7-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-4-(4H-1,2,4-triazol-3-yl)piperidine
3-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-1,5,6-trimethyl-1,2-dihydropyridin-2-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-2-methoxy-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}acetamide
N-methyl-N-(oxan-2-ylmethyl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
3-[(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-1-(cyclobutylmethyl)-3-hydroxypiperidin-2-one
(2S)-2-amino-3-(1H-imidazol-4-yl)-N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}propanamide
methyl 2-(5-methyl-2-{[2-(pyridin-4-ylsulfanyl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
2-benzyl-4-[3-(3-methylphenoxy)azetidine-1-carbonyl]-1,3-thiazole
1-(oxane-4-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
N-[2-(2-methoxyphenyl)ethyl]-2-(4-{4-[(oxan-4-yl)amino]piperidin-1-yl}phenyl)acetamide
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-[(3E)-4-methylhex-3-en-1-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]pyrimidin-4-amine
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(3-methoxyphenoxymethyl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
2-(2-hydroxyethyl)-8-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
4-methyl-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)-1,3-oxazole-5-carboxamide
4-phenyl-5-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazole
3-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-(trifluoromethyl)morpholin-4-yl]quinoline
1-[(3-chlorophenyl)methyl]-3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine
N-(2-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-oxoethyl)methanesulfonamide
1-[(2,4-difluorophenyl)methyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one