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N-(4-carbamoyl-3-chlorophenyl)-4-phenylazepane-1-carboxamide
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}acetamide
5-[(E)-2-phenylethenyl]-1H-indazol-3-amine
5-methanesulfonyl-4-(piperidin-3-yl)-2-(pyridin-2-yl)pyrimidine
2-[(2,4,5-trimethylphenyl)methyl]-2,7-diazaspiro[4.5]decane
3-(pyrrolidine-1-carbonyl)-1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidine
2-[1-(2,3-dihydro-1H-inden-2-yl)-5-[4-(methoxymethyl)-5-methyl-1,2-oxazol-3-yl]-1H-1,2,4-triazol-3-yl]acetamide
5-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-1,2-dihydropyridin-2-one
2-(4-hydroxyphenyl)-1-(2-methyl-4-phenylpiperazin-1-yl)ethan-1-one
2-[(3-methoxyphenyl)methyl]-8-[2-(methylsulfanyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2-{1-[(2-fluorophenyl)methyl]-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-methyl-N-[1-(pyridin-2-yl)propan-2-yl]acetamide
N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carboxamide
3-(2-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-2-methoxy-N-(oxolan-2-ylmethyl)pyridine-3-carboxamide
1-benzyl-5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-N-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
(2S,4R)-4-amino-1-(4-cyclohexylbutanoyl)-N-ethylpyrrolidine-2-carboxamide
N-(2-hydroxyethyl)-2-(pyrrolidin-1-yl)-N-(1,3-thiazol-2-ylmethyl)benzamide
2-{[6-(4-cyclohexylpiperazin-1-yl)pyridazin-3-yl]oxy}-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
N-cyclohexyl-1,5-dimethyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
N-methyl-2-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carboxamide
4-methyl-N-[5-(4-methylphenoxymethyl)-1,3,4-thiadiazol-2-yl]-3-oxopiperazine-1-carboxamide
6-(benzyloxy)-4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-4-(2-oxopiperidin-1-yl)butanamide
4-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-6-fluoro-1,2-dihydroquinolin-2-one
N-cyclopropyl-2-(pyridin-3-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
6-[(3,4-difluorophenyl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
(3aR,6aR)-2-cyclobutanecarbonyl-5-(5-propyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(2-fluorophenoxy)ethyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
N,4-dimethyl-6-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-2-amine
1-ethyl-4-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonane-7-carbonyl]-1,2-dihydropyridin-2-one
2-({[3-hydroxy-2-oxo-1-(3-phenylpropyl)piperidin-3-yl]methyl}(methyl)amino)-N-methylacetamide
(2S,4R)-1-benzyl-N-(2-methoxyethyl)-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)amine
N-[1-(4-chlorophenyl)ethyl]-5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
1-[2-(dimethylamino)-4-{[3-(propan-2-yloxy)propyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-{[2-(dimethylamino)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]thiophene-2-carboxamide
1-({5-[1-(3-ethyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
N-{[3-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-{2-[cyclohexyl(methyl)amino]ethyl}-8-(2-hydroxyacetyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[3-cyclopropyl-5-(2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}ethyl)-1H-1,2,4-triazol-1-yl]pyridine
4-methoxy-6-(5-methyl-1H-indol-3-yl)pyrimidin-2-amine
N-[3-(cyclopentyloxy)propyl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
3-[(3-chlorophenyl)methyl]-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[3-(1H-imidazol-1-yl)propanoyl]-4-(2-methylphenoxy)piperidine-4-carboxylic acid
1-(1-ethylpyrrolidine-3-carbonyl)-4-(4-methoxybenzoyl)piperazine
2-methyl-5-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
4-[(2-methyl-5-oxo-4-phenylpiperazin-1-yl)sulfonyl]benzoic acid
5-(2-phenylethyl)-5-(1-{[4-(pyrrolidin-1-yl)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione