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3-[(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-7-fluoro-1-(oxolan-2-ylmethyl)-1,2-dihydroquinolin-2-one
5-chloro-N,4,6-trimethyl-2-oxo-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydropyridine-3-carboxamide
6-[(diethylamino)methyl]-N-(2-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N'-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-N-methylbutanediamide
4-{[1-(2,6-dimethylquinoline-4-carbonyl)azetidin-3-yl]oxy}benzoic acid
3-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1-[2-(propan-2-ylsulfanyl)phenyl]urea
methyl 3-{[4-(3-hydroxyphenyl)piperazine-1-carbonyl]amino}-4-methylbenzoate
2-methoxy-4-(1-{2-[(1-methylpiperidin-4-yl)oxy]phenyl}-1H-imidazol-2-yl)phenol
(1R,3S)-3-(2-hydroxyethoxy)-7-[(3-methylpyrazin-2-yl)methyl]-7-azaspiro[3.5]nonan-1-ol
[(2-chloro-6-fluorophenyl)methyl](ethyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
2-[1-(cyclopropylmethyl)-4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-2-yl]ethan-1-ol
3-(4-methyl-1,3-thiazol-5-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}propanamide
ethyl 1-({6-methyl-1-[(2-methylphenyl)methyl]-2-oxo-1,2-dihydroquinolin-3-yl}methyl)piperidine-4-carboxylate
1-cyclohexyl-4-(2-ethylpyrimidine-5-carbonyl)-1,4-diazepane
N-(1-cycloheptylpiperidin-3-yl)-5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
3-fluoro-N-(1-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
2,2-dimethyl-5-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}thiomorpholin-3-one
N-[4-(2-fluorophenoxy)phenyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxamide
6-methyl-2-{[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]amino}pyridine-3-carboxamide
2-[(4aR,7aS)-4-(1-ethyl-1H-pyrazole-5-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,3,4-trimethoxybenzamide
N-[(2-chlorophenyl)methyl]-2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
N,N-diethyl-2-{[4-(2-methoxypyridine-3-carbonyl)-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl]oxy}acetamide
3-[2-(3-methoxyphenoxy)ethyl]-4-methylbenzamide
3-{1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]piperidin-3-yl}benzoic acid
ethyl 1-(5-acetylthiophene-3-carbonyl)-3-[(3-chlorophenyl)methyl]piperidine-3-carboxylate
1-(2-phenoxyethyl)-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperazine
(3-benzyl-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-yl)methanol
2-(cyclohexylmethyl)-4-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}morpholine
N-ethyl-3-methyl-3,9-diazaspiro[5.6]dodecane-9-carboxamide
1-cyclohexyl-N5-cyclopropyl-N3-(cyclopropylmethyl)-4-oxo-N3-propyl-1,4-dihydropyridine-3,5-dicarboxamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-(cyclopropylmethyl)-9-(2-hydroxy-5-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 2-amino-3-cyano-4-(5-cyano-1-methyl-1H-pyrrol-3-yl)-5,6,7,8-tetrahydroquinoline-6-carboxylate
N-(1-{7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
N-[(2R,3R)-1'-[(2,4-difluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
4-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)pyridine
3-phenoxy-1-[2-(piperidin-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
1-methyl-9-[2-(methylamino)benzoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
1-(furan-2-yl)-2-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethane-1,2-dione
5-[4-(1H-imidazol-1-yl)butanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
N-[(3S,4R)-1-[2-(5-acetylthiophen-3-yl)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
5-(1-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-3-methyl-1H-1,2,4-triazole
[(6-methoxy-2H-chromen-3-yl)methyl](methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
(4aS,7aR)-1-(5-methyl-1,2-oxazole-3-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2R,3R)-3-({1-[(3-methylphenyl)methyl]cyclopropyl}amino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(1r,4r)-4-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)cyclohexan-1-ol
4-[1-(2-methylphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]-1λ6-thiane-1,1-dione