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3-butanamido-N-(1-propylpiperidin-3-yl)benzamide
N-[2-(dimethylamino)ethyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-(1-{7-[(2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-5-(methoxymethyl)furan-2-carboxamide
N,N-dimethyl-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
4-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-methylpiperazine-2-carboxylic acid
N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}oxane-4-carboxamide
(1R,5R)-6-benzyl-3-(2-ethoxypyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(1H-indole-2-carbonyl)-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
3-[2-(4-fluorophenyl)ethyl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
1-[3-(azetidine-1-carbonyl)benzenesulfonyl]-N-methylpiperidine-2-carboxamide
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-methoxyphenyl)-2-methylpiperazine
3-(2H-1,3-benzodioxol-5-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
4-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-(2-chlorobenzoyl)piperidine
3-[1-(cyclopropanesulfonyl)piperidin-3-yl]-1-[2-(dimethylamino)ethyl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-N-methylbenzene-1-sulfonamide
5-[2-amino-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1H-1,2,4-triazol-3-amine
N-(3-methoxypropyl)-1-methyl-5-[4-(pyrrolidin-1-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
ethyl 1-[2-(2-phenylethyl)-1,3-benzoxazole-5-carbonyl]piperidine-3-carboxylate
N-{1-[(4-methylphenyl)methyl]cyclopropyl}morpholine-2-carboxamide
N-phenyl-2-{[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]amino}butanamide
3-[1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
2-cyclopropyl-8-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
N-cyclopentyl-N-[(2-methylphenyl)methyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
3-[1-(butan-2-yl)-1H-pyrazol-5-yl]-1-[(4-chlorophenyl)methyl]-1-(3-hydroxypropyl)urea
2-[(3-chlorophenyl)methyl]-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,3-benzoxazole-6-carboxamide
3-[(dimethylamino)methyl]-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)pyrrolidin-3-ol
8-chloro-2-{[(pyridin-3-ylmethyl)amino]methyl}quinolin-4-ol
N,N-dimethyl-1-{2-[(4-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}pyrrolidine-2-carboxamide
methyl 2-(1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
2-[1-methyl-4-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperazin-2-yl]ethan-1-ol
N-ethyl-N-[1-(4-methoxyphenyl)propyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
2-methyl-3-[5-(3-methylfuran-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-6-(trifluoromethyl)pyridine
methyl 3-[(4-{2-[3-(morpholin-4-ylmethyl)phenoxy]ethyl}piperazin-1-yl)sulfonyl]thiophene-2-carboxylate
3-amino-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}pyrrolidine-3-carboxylic acid
2-methyl-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
5-(2-{4-[benzyl(methyl)amino]piperidin-1-yl}-2-oxoethyl)-1,3-dimethylimidazolidine-2,4-dione
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(2,5-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
3-(4-ethyl-1H-pyrazol-5-yl)-1-[3-(2-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidine
4-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(pyrrolidin-1-yl)-6-(trifluoromethyl)pyrimidine
3-[1-(2-phenoxyacetyl)piperidin-3-yl]benzoic acid
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(2,3-difluorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-2-(ethylamino)pyrimidine-5-carboxamide
2-fluoro-N-[2-hydroxy-2-(3-methoxyphenyl)ethyl]-5-sulfamoylbenzamide
(4aS,7aR)-1-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(1,2-oxazol-3-ylmethyl)-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
5-[2-(2-methyl-1H-indol-3-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
8-(1H-1,2,3-benzotriazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N,1-dimethylpyrrolidin-3-amine