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N-[2-(2-chlorophenyl)-1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-(thiophen-3-ylmethyl)furan-2-carboxamide
N-({1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}methyl)-2,3-dihydro-1H-indene-2-carboxamide
1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carbonyl)azetidin-3-ol
3-(pyridin-3-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
3-({4-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]piperidin-1-yl}methyl)pyridine
1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-[4-(4-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]urea
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
8-(1H-indol-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4S)-N-ethyl-4-(2-fluoro-6-methoxybenzamido)-1-(pent-2-yn-1-yl)pyrrolidine-2-carboxamide
3-methoxy-N-methyl-4-[(1-methylpiperidin-4-yl)oxy]-N-[2-(oxan-4-yl)ethyl]benzamide
6-chloro-N,1-dimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-indole-2-carboxamide
8-(2-hydroxyacetyl)-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(3-fluorophenoxy)-1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]azetidine
N-[(2S,4R,6S)-2-(4-methoxy-3-methylphenyl)-6-(2-phenylethyl)oxan-4-yl]acetamide
3-ethoxy-N-[3-(2-hydroxyphenyl)propyl]-4-(prop-2-en-1-yloxy)benzamide
N-[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]pyrimidin-2-amine
2-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
1-ethyl-N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-6-oxopiperidine-3-carboxamide
5-({3-[3-(3-chlorophenyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)isoquinoline
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(2-methyl-1H-imidazol-1-yl)propanamide
N-cyclopropyl-N-(2-phenyl-1-{1-[(2,3,6-trifluorophenyl)methyl]piperidin-4-yl}ethyl)pyridine-2-carboxamide
5-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]pyridine-2,4-diol
N-{2-[2-(trifluoromethoxy)phenyl]ethyl}-1H-1,2,3-triazole-5-carboxamide
4-(1H-imidazol-2-yl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
5-[2-(3-chlorophenoxymethyl)pyrimidin-4-yl]-2-ethoxybenzoic acid
[(3R,4R)-1-(4-methoxyquinoline-2-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-(2-methoxyethyl)-1-[1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
N-({1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-dichlorobenzamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-4-(4-methyl-1H-pyrazol-3-yl)piperidine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-4-(1H-imidazol-1-yl)-N-methylbenzamide
1-(morpholin-4-yl)-3-[1-(4-propylpyrimidine-5-carbonyl)piperidin-4-yl]propan-1-one
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N,N-bis(pyridin-3-ylmethyl)acetamide
8-(2,2-dimethylpropyl)-1-ethyl-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3S,5S)-1-cyclopentyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(cyclopropylmethyl)-4-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-2-(propan-2-yl)-1,4-diazepane
(3S,4S)-1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-4-propylpyrrolidine-3-carboxylic acid
2-(4-{[3-(2-hydroxyethyl)-4-(2-phenylethyl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
3-[(cyclopropylamino)methyl]-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
4-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-6-methyl-1,2-dihydroquinolin-2-one
4-[2-(propan-2-ylsulfanyl)ethyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-[(3-methoxyphenyl)sulfanyl]-N-methylacetamide
3-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1-methyl-1H-indole
1-[(3-ethoxy-4-hydroxyphenyl)methyl]-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-4-methoxy-N-(oxolan-2-ylmethyl)pyridine-2-carboxamide
9-(3,4-dimethylbenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
{3-[(3-chlorophenyl)methyl]-1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-yl}methanol