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1-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2-methyl-2-(thiophen-2-ylformamido)propanamide
N,N-diethyl-1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidine-3-carboxamide
methyl (2S)-1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxylate
N-[4-(2,2-dimethylpropanamido)-3-methoxyphenyl]-2,6-dimethoxypyrimidine-4-carboxamide
3-(3-hydroxyquinoxalin-2-yl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
6-methyl-4-oxo-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-4H-pyran-2-carboxamide
N,5-dimethyl-N-[2-(oxan-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
2-{[4-(naphthalen-1-yl)-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(1-{2-[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}piperidin-2-yl)methanol
N-(1-butyl-3-methyl-1H-pyrazol-5-yl)-4-hydroxy-4-phenylpiperidine-1-carboxamide
1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetamide
1'-({5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-(2-methoxyethyl)-N-methyl-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-amine
(2S,4R)-4-({[4-(benzyloxy)phenyl]methyl}amino)-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-3-phenoxypropanamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-[4-(trifluoromethyl)phenyl]ethan-1-one
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(2,3,4-trifluorophenyl)ethan-1-one
3-[4-(benzyloxy)piperidine-1-carbonyl]-1H-indazole
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropane-1-carboxamide
2-amino-N-{2-[(E)-2-phenylethenyl]phenyl}acetamide
1-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
1-benzyl-5-cyclopentyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
N-(2-methoxyethyl)-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-[4-(5-aminopyridin-3-yl)phenyl]-3,3-diethylurea
2-{2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
methyl[(2-phenyl-1,3-oxazol-4-yl)methyl][2-(pyridin-4-yl)ethyl]amine
[2,4,6-trimethyl-3-({[2-(pyrrolidine-1-sulfonyl)ethyl]amino}methyl)phenyl]methanol
(1s,4s)-N-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexan-1-amine
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-methoxyacetamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(morpholine-4-carbonyl)pyrrolidin-3-yl]acetamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)cyclopentanecarboxamide
N-methyl-2-(pyridin-2-ylsulfanyl)-N-(thiophen-3-ylmethyl)propanamide
2-cyclopropyl-8-[(5-ethylpyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-1-yl)ethan-1-ol
N-(3-methyl-1-{7-[(4-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
6-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-{7-[ethoxy(phenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-4-phenylbutane-1,4-dione
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-(pyridin-2-ylmethyl)propanamide
3-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-N-methylpropanamide
4-(pentan-3-yl)-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
5-{3-oxo-3-[4-(quinazolin-2-yl)piperazin-1-yl]propyl}-5-(thiophen-2-ylmethyl)pyrrolidin-2-one
3-(3,4-dimethylphenyl)-4-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}-1H-pyrazole
2-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one