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N-{[2-(diethylamino)pyridin-3-yl]methyl}-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
(1-{[2-(difluoromethoxy)phenyl]methyl}azepan-2-yl)methanol
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-(2-oxopyrrolidin-3-yl)benzamide
2-{1-benzyl-5-[2-(2-oxoazepan-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}acetamide
1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2-(1,3-thiazol-2-yl)piperidine
2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)acetamide
(3R,4R)-1-(6-aminopyridine-3-carbonyl)-3-cyclopropyl-4-methylpyrrolidin-3-ol
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
methyl 3-(2-methylbenzoyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-methyl-1-[2-(methylsulfanyl)phenyl]-4-{2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetyl}piperazin-2-one
4-(4-{3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidine-1-carbonyl}phenyl)-2-methylbut-3-yn-2-ol
N-(1-benzylpiperidin-3-yl)-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
4,6-dimethyl-2-[3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carbonitrile
N-({7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1H-1,3-benzodiazole-5-carboxamide
N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
4-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}benzonitrile
2-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)benzene-1,3-diol
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-N'-(2-fluoro-5-methylphenyl)butanediamide
7-chloro-2-methyl-4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(5-chlorothiophen-2-yl)methyl]-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanamide
3-[(2-fluorophenyl)methyl]-1-methyl-6-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-(2-methoxyphenoxy)-1-{2-methylthieno[3,2-d]pyrimidin-4-yl}azetidine
7-cyclohexyl-2-(3-hydroxypyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-4-(1,2,3,4-tetrahydroisoquinolin-7-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-{[3-(2-aminoethyl)piperidin-1-yl]methyl}-6-methylquinolin-4-ol
ethyl 2-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)acetate
N-[(2-phenoxypyridin-3-yl)methyl]cyclobutanecarboxamide
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2-(1H-pyrazol-1-yl)benzamide
3-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydroisoquinolin-1-one
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1,9-dioxaspiro[5.5]undecan-4-amine
N-[2-(furan-2-yl)ethyl]-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(3-hydroxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(3-fluoro-4-methoxyphenyl)methyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[2-(thiophen-2-yl)azetidin-1-yl]ethan-1-one
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)(pyridin-2-ylmethyl)amine
N-[(2R,3R)-1'-(3,5-difluorobenzoyl)-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
(3aR,5S,6S,7aS)-2-{[5-(oxan-2-yl)furan-2-yl]methyl}-octahydro-1H-isoindole-5,6-diol
2-{4-[(3-fluorophenyl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
[1-(3-{[2-(2-aminoethyl)quinazolin-4-yl]amino}propyl)piperidin-3-yl]methanol
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
({2-[(2-chloroprop-2-en-1-yl)oxy]-7-(methylsulfanyl)quinolin-3-yl}methyl)[(5-methylpyrazin-2-yl)methyl]amine
1-{[(3R,4R)-1-(furan-3-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
4-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenol
9-(cyclohex-3-ene-1-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
3-(3-hydroxy-3-methylbutyl)-N-(5-methylhexan-2-yl)benzamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
1-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-methyl-1,2-dihydroquinoxalin-2-one