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4-methyl-5-(1-phenyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-amine
N-(1-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-2-fluorobenzamide
2-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-N,N-dimethylpyridine-3-carboxamide
3-ethyl-N,N-bis(2-hydroxyethyl)-1H-indole-2-carboxamide
6-cyclopentyl-1-methyl-N-[(1-propylpiperidin-3-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(3S,4S)-3-hydroxy-4-[methyl(propyl)amino]pyrrolidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-methyl-2-phenylpropan-1-one
{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[3-(methylsulfanyl)propyl]amine
7-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}sulfonyl)-2,7-diazaspiro[4.5]decane
7-(5-chloropyridin-2-yl)-4-(6-methylpyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidin-4-ol
N,N-dimethyl-2-(4-methyl-3-phenylpiperazine-1-carbonyl)aniline
[1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl](thiophen-2-yl)methanol
2-[4-(4-chlorophenyl)-2-methyl-5-oxopiperazin-1-yl]acetic acid
2-(ethylamino)-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}pyrimidine-5-carboxamide
1-(2-aminoethyl)-N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-1H-1,2,3-triazole-4-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(1-fluoro-3-phenylpropan-2-yl)acetamide
N,N-dimethyl-1-{4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}methanesulfonamide
3-(3-{furo[3,2-c]pyridin-4-yl}phenyl)-1-(pyrrolidin-3-ylmethyl)-1H-pyrazole
5-acetyl-N-[1-({[(4-phenyloxan-4-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]thiophene-2-carboxamide
5-[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]pyridine-2-carbonitrile
3-(1-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-4-phenyl-1H-imidazol-5-yl)benzonitrile
N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-1,2,5-thiadiazole-3-carboxamide
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-4-(3-fluorophenoxy)piperidine
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]amine
2-[(5-methylpyrazin-2-yl)methyl]-8-(6-methylpyridine-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-ethoxy-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
2-[(5-methylpyrazin-2-yl)methyl]-9-[(6-methylpyridin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(4-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}piperazin-1-yl)quinazoline
3-methoxy-N-(1-{7-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
5-(azocane-1-carbonyl)-2-methyl-1H-1,3-benzodiazole
1-(2-{[2-(diethylamino)ethyl]amino}pyrimidin-4-yl)piperidin-3-ol
3-{2-[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,4-triazol-5-amine
1-[(3-methylpyridin-2-yl)methyl]-4-(1,3-thiazol-2-ylmethyl)piperazine
N-[(4-fluoro-2-methoxyphenyl)methyl]-7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
4-{3,9-diazaspiro[5.6]dodecan-9-yl}-N-(4-methylpyridin-2-yl)-4-oxobutanamide
5-(azocane-1-carbonyl)-N-ethylpyrimidin-2-amine
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
(3S,4R)-1-(morpholine-4-sulfonyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
3-fluoro-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzene-1-sulfonamide
N-[2-(dimethylamino)ethyl]-1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
2-(dimethylamino)-7-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-methyl-N-{4-[(3E)-pent-3-enamido]phenyl}benzamide
1-(cyclohexylmethyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
3-{[(4-fluorophenyl)methyl]sulfanyl}-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
methyl 4-[6-amino-5-cyano-4-(3-ethyl-1H-pyrazol-5-yl)pyridin-2-yl]-5-methylfuran-2-carboxylate
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(3-phenyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methanol
2-(propan-2-yl)-9-[4-(1H-pyrazol-3-yl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-1-(1-cyclobutanecarbonylpiperidin-4-yl)-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
5-cyclopentyl-3-{[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]methyl}-1,2,4-oxadiazole