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N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3-fluoroimidazo[1,2-a]pyridine-2-carboxamide
4-[1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3-carbonyl]morpholine
(3S)-3-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]azepan-2-one
2-(2-butyl-1H-imidazol-4-yl)-1-(furan-3-ylmethyl)-1H-imidazole
(1R,3S)-3-methoxy-7-[4-(trifluoromethyl)pyrimidin-2-yl]-7-azaspiro[3.5]nonan-1-ol
N-{2-[5-(4-hydroxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}propanamide
4-(3-fluoropyridin-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[6-(morpholin-4-yl)pyridine-3-carbonyl]-4-phenylazepane
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-5-(hydroxymethyl)furan-2-carboxamide
3-(morpholine-4-sulfonyl)-5-(4-phenyl-1H-imidazol-1-yl)benzoic acid
5-(2-methylpropyl)-1'-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-methoxy-N-[1-methyl-7-(2-methyl-4-phenylpiperazine-1-carbonyl)-2-(pyridin-4-yl)-1H-1,3-benzodiazol-5-yl]acetamide
8-[2-(azepan-1-yl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-1-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]urea
2-[(4-ethoxyphenyl)methyl]-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
8-(3-cyano-2-methoxypyridin-4-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(4aS,7aR)-N-(2-fluorophenyl)-6,6-dioxo-4-pentyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
ethyl 4-benzyl-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidine-4-carboxylate
2-[methyl(pyridin-3-ylmethyl)amino]-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}acetamide
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl})amine
4-[7-(carbamoylcarbonyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
7-[4-(pyridin-2-yl)pyrimidin-2-yl]-2,7-diazaspiro[4.5]decane
2-amino-7-(3-ethyl-5-hydroxyadamantane-1-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(methanesulfonylmethyl)piperidine
N-ethyl-5-(2-fluorophenoxymethyl)-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1H-pyrazole-3-carboxamide
2-[(4-methylpiperazin-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-(1-{1-[4-(piperidin-1-yl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
methyl (2S,4S,5R)-5-(3-chlorophenyl)-1-methyl-4-{[(2-methyl-1,3-thiazol-4-yl)methyl]carbamoyl}pyrrolidine-2-carboxylate
2-(3-{[5-(4-methylphenyl)-1H-pyrazol-3-yl]formamido}propanamido)acetic acid
1-(2,4,6-trimethyl-3-{[2-(trifluoromethyl)morpholin-4-yl]methyl}phenyl)ethan-1-one
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-[4-(2-propyl-1H-imidazol-1-yl)phenyl]ethan-1-ol
N-(1-methanesulfonylpiperidin-4-yl)-2-(1H-1,2,4-triazol-3-yl)benzamide
N-tert-butyl-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[1-(7-{[3-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-3-methylbutyl]acetamide
N-(1-{7-[(2,6-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)propanamide
4-[4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazine-1-carbonyl]morpholine
8-(4-aminopyrimidin-2-yl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[1-(2H-1,3-benzodioxol-5-ylmethyl)-4-hydroxypiperidin-4-yl]-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
5-acetyl-N-[2-(1-ethylpiperidin-3-yl)ethyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
ethyl 1-{[4-(methylsulfanyl)phenyl]carbamoyl}-4-(2-phenylethyl)piperidine-4-carboxylate
(1R,3S)-3-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]cyclopentan-1-amine
N-(1-{7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxybenzamide
methyl 6-[(benzylsulfamoyl)amino]-1,2,3,4-tetrahydroquinoline-1-carboxylate
N-cyclobutyl-3-{[(1R,2S)-2-(methoxymethyl)cyclopentyl]sulfamoyl}benzamide
(1S,5R)-N-(3-methoxyphenyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-({5-[1-(furan-2-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)azepane
2-{4-[(2-chloro-4-fluorophenyl)methyl]-1-(2,2-dimethylpropyl)piperazin-2-yl}ethan-1-ol
4-{[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]methyl}benzonitrile