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5,6-dimethyl-2-oxo-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyrrolidin-1-yl)benzamide
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
3-amino-1-{4-[4-(propan-2-yl)-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}propan-1-one
2-[(2-chlorophenyl)methyl]-4-(piperidine-1-sulfonyl)morpholine
2-[bis(prop-2-en-1-yl)amino]-2-(4-fluoro-3-methylphenyl)acetic acid
N-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-2-(pyridin-3-yl)piperidine-1-carboxamide
3-[1-(2-fluorophenyl)piperidin-4-yl]-1-[3-(2-methoxyethoxy)phenyl]urea
1-{2-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}ethan-1-one
3-[(3S,4R)-1-benzyl-4-(4-methylpiperazin-1-yl)piperidin-3-yl]-N-[3-(methylsulfanyl)phenyl]propanamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[methyl(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
1-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
6-[(4-hydroxy-4-methylazepan-1-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
1-[(3R)-3-cyclopropyl-3-hydroxy-4,4-dimethylpyrrolidin-1-yl]-2-(methylsulfanyl)ethan-1-one
1-[2-methoxy-5-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
2-(azepan-1-yl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(2-methylpyrimidin-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(1S,5R)-3-[(3-chloro-4-fluorophenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(pyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)piperidine-1-carboxamide
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(4-methoxybenzoyl)piperidine
N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
3-[2-(4-cyclopentylpiperazin-1-yl)-2-oxoethyl]-1-cyclopropyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
N-(furan-2-ylmethyl)-N,1-dimethyl-5-[(2-phenylethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-tert-butyl-5-[1-(methoxymethyl)cyclopropyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl){[2-(1H-pyrazol-1-yl)phenyl]methyl}amine
3-[2-(4-methoxyphenyl)ethyl]-1-(thiophene-3-carbonyl)piperidine
3-(4-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)propanamide
1-{1-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]cyclopentyl}pyrrolidine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-propyl-1,2-oxazole-4-carboxamide
N-{2-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
methyl 3-{[4-(3-methylthiophene-2-carbonyl)-7-oxo-1,4-diazepan-1-yl]methyl}benzoate
1-(2,3-dimethylphenyl)-N-{[3-(methylsulfanyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-({7-[(3,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2,5-dimethylfuran-3-carboxamide
N5-(prop-2-en-1-yl)-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
5-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
5-(2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one
N-(furan-2-ylmethyl)-3-(3-methyl-1H-pyrazol-1-yl)-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}propanamide
2-(3-methoxypropyl)-1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}piperidine
2-(furan-2-yl)-4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[3-(4-methylpiperazin-1-yl)propyl]piperidin-2-one
1-(3-phenylpropyl)-N-{[2-(trifluoromethoxy)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-[1-(1H-pyrazole-4-carbonyl)piperidin-4-yl]morpholine
N-[2-({1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)ethyl]acetamide
N-(1-hydroxybutan-2-yl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-{2-[1-(1-acetyl-1,2,3,4-tetrahydroquinolin-6-yl)-1H-imidazol-4-yl]ethyl}acetamide
2-{[4-(3-methoxyphenyl)-5-(3-methylthiophen-2-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
ethyl 4-(3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamido)piperidine-1-carboxylate
(3S,4S)-1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3,4-diol
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one