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N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-2-(morpholin-3-yl)acetamide
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-4-(pyridin-3-yl)pyrimidin-2-amine
4-hydroxy-2-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}quinoline-6-carboxamide
3-[({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)carbamoyl]pyridin-1-ium-1-olate
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(quinazolin-4-yloxy)acetamide
3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)-5-[1-(3-phenylpropanoyl)piperidin-4-yl]imidazolidine-2,4-dione
5-benzyl-5-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
7-chloro-N,N-dimethyl-2-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
5-[({[3-(cyclopentyloxy)phenyl]carbamoyl}amino)methyl]-N-methylfuran-2-carboxamide
methyl({[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})(pyrazin-2-ylmethyl)amine
2,6-difluoro-N-({7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
4-({5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}methyl)benzene-1-sulfonamide
2-(2,4-dimethylphenyl)-1H-1,3-benzodiazole-6-carboxylic acid
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methyl-N-(1,3-thiazol-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
2-{[(adamantan-1-yl)amino]methyl}-4-(2,5-dimethoxyphenyl)phenol
4'-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-[(4-chlorophenyl)methyl]-5-{3-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-3-oxopropyl}pyrrolidin-2-one
5-({5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}methyl)-3-(2-phenylethyl)-1H-1,2,4-triazole
methyl 4-({4-[1-(2,3-dihydro-1H-inden-2-yl)-4-methyl-2,5-dioxoimidazolidin-4-yl]piperidin-1-yl}methyl)benzoate
2-hydroxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-4-(methylsulfanyl)butanamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
7-(1-benzothiophen-3-yl)-9-(pyridin-2-ylmethoxy)-4-(1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{[(1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)oxy]methyl}pyridine
[3-(3-methoxypropyl)-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-3-yl]methanol
methyl 2-(3-{3-[5-(dimethylcarbamoyl)furan-2-yl]phenyl}-1H-pyrazol-1-yl)propanoate
2-(4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-1-[(2-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
1-(cyclohexylmethyl)-5-[4-(hydroxymethyl)piperidin-1-yl]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
[1-(1-methylpiperidine-2-carbonyl)-4-(2-phenylethyl)piperidin-4-yl]methanol
5-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
[(4,5-dimethylfuran-2-yl)methyl][2-methoxy-1-(pyridin-2-yl)ethyl]methylamine
5-methyl-6-(4H-1,2,4-triazol-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-[2-(3-fluorophenyl)ethyl]-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)urea
N,2-dimethyl-N-(oxan-2-ylmethyl)-2-phenylpropanamide
5-methoxy-3-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}-1H-indazole
3-[3-(pyridin-2-yl)azetidine-1-carbonyl]-5,6,7,8-tetrahydroquinoline
2-methyl-6-(2-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)pyridine
methyl 4-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}benzoate
1-cyclopentyl-4-{5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carbonyl}piperazine
(5S,9aS,9bS)-2-cyclopentyl-5-(5-methylfuran-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-{1-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]piperidin-4-yl}-3-[(4-fluorophenyl)methyl]-5-methylimidazolidine-2,4-dione
2-[(4-methylpiperidin-1-yl)methyl]-4-phenylphenol
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(thiophen-2-yl)propan-2-yl]benzamide
benzyl({[3-(2,2-diethylmorpholine-4-carbonyl)-1,2-oxazol-5-yl]methyl})methylamine
benzyl({[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl})(cyclopropylmethyl)amine
N-(2-methoxyethyl)-3-(1H-pyrazol-4-yl)-N-(thiophen-3-ylmethyl)benzamide
1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-1,4-diazepane-6-carboxylic acid