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4-(cyclopropylmethyl)-2-[(3-fluorophenyl)methyl]morpholine
N-cyclohexyl-4-hydroxy-N-(2-hydroxy-2-phenylethyl)-2-methylpyrimidine-5-carboxamide
2-[(1S,5S)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1H-1,3-benzodiazole
4-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}-5-phenyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-2-one
3-{[(cyclohexylmethyl)amino]methyl}-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
2-[methyl(2-phenylethyl)amino]-N-(1-methyl-2-oxopyrrolidin-3-yl)-2,3-dihydro-1H-indene-2-carboxamide
4-(1-ethyl-1H-imidazol-2-yl)-N-(2-fluorophenyl)piperidine-1-carboxamide
3-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
methyl 5-(3-{2-[(4-methoxy-2-methylphenyl)carbamoyl]ethyl}piperidin-1-yl)-5-oxopentanoate
1-methyl-4-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperazine
2-{1-ethyl-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
N-(1-benzylpyrrolidin-3-yl)-3-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}propanamide
4-[3-(2-methoxyethyl)-5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
N-[4-(pyridin-3-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]pyrrolidine-1-carboxamide
6-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}-1,2-dihydroisoquinolin-1-one
4-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-N,N-dimethyl-4-oxobutanamide
N3-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-N5-[(3,4,5-trifluorophenyl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-(2,3-difluoro-6-methoxyphenyl)-1-(2-methanesulfonylethyl)-1H-imidazole
ethyl 4-{2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
N-[(2-chloropyridin-3-yl)methyl]-N-methyl-2-(methylamino)benzamide
1-cyclohexyl-N-[(3,4,5-trimethoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
methyl 3-(1H-indol-2-ylmethyl)-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1S,5R)-6-(cyclobutylmethyl)-3-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]-N-[2-(2-methoxyphenyl)ethyl]acetamide
[1-(4-methylphenyl)propan-2-yl]({1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
2-methoxy-3-[2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]quinoline
{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
5-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
5-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]thiophene-2-carboxamide
methyl 3-[(3S,4R)-1-[(4-methoxynaphthalen-1-yl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
3-[(3R,4S)-1-(4-chloro-2-methoxybenzoyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
[1-(cyclohex-1-ene-1-carbonyl)-3-[(2,4-difluorophenyl)methyl]piperidin-3-yl]methanol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
1-[2-({[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-3-ol
N-[(2-chloro-6-fluorophenyl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
3-({5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)-2,2-dimethylpropan-1-ol
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-1,1-dioxo-1λ6-thiolane-3-carboxamide
3-[4-(dimethylcarbamoyl)phenyl]-5-(morpholine-4-sulfonyl)benzoic acid
4-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
2-{2-[5-(2-chlorophenyl)furan-2-yl]-1H-imidazol-1-yl}ethan-1-ol
2-methoxy-N-[1-(3-phenylpropyl)piperidin-3-yl]pyridine-3-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
2-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
(1R,2R,6S,7S)-N-(8-chloroquinolin-5-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
N-(2-methoxyethyl)-2-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-1,4-dihydroquinoline-8-carboxamide
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-(naphthalene-1-carbonyl)piperidine
1-[2-(dimethylamino)ethyl]-3-(3-methoxyphenyl)-3-[2-(4-methyl-3-phenylpiperazin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
methyl 4-[({[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]benzoate
5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
N-({7-[2-(3,4-difluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-methoxy-2-phenylacetamide