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1-methyl-5-(4-methyl-1,4-diazepane-1-carbonyl)-2-(morpholin-4-yl)-1H-1,3-benzodiazole
2-(4-methanesulfonylphenyl)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
1-{1-oxa-8-azaspiro[4.5]decan-8-yl}-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
2-[(trimethyl-1H-pyrazol-1-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
ethyl 4-[(4-{[1-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
2-(dimethylamino)-N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-4-methylpyrimidine-5-carboxamide
2-(5-acetamido-1H-1,2,4-triazol-3-yl)-N-ethyl-N-[2-(3-methylphenoxy)ethyl]acetamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(4H-1,2,4-triazol-4-yl)propanamide
2-(1-benzothiophen-7-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-(2-methylpropyl)-5-[1-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazole
(2R,3R,6R)-3-(4-fluorophenyl)-5-(5-methyl-1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N4-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-5-ethylpyrimidine-2,4-diamine
1-[3-(3-chlorophenyl)-3-phenylpropanoyl]piperidine-4-carboxamide
4-({1-[(4-fluorophenyl)methyl]-5-(1H-1,2,3,4-tetrazol-1-ylmethyl)-1H-1,2,4-triazol-3-yl}methyl)-1-methylpiperidine
1-cycloheptyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2,4-difluoro-N-(pyridin-3-ylmethyl)benzamide
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(2-methyl-1,3-thiazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2,1,3-benzoxadiazol-4-ylmethyl)[(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amine
6-ethyl-N-[(4-fluorophenyl)methyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
1-[4-(4-ethoxy-3-methylphenyl)-4-oxobutanoyl]piperidine-4-carboxylic acid
4-(4-acetamido-1H-pyrazol-1-yl)-N-(thiophen-3-ylmethyl)benzamide
1-(2,3-dihydro-1H-inden-5-yl)-3-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]urea
N-(3-ethoxypropyl)-4-(piperidin-3-yl)benzamide
4-hydroxy-1-(3-methylfuran-2-carbonyl)piperidine-4-carboxylic acid
ethyl 1-(1-benzylpyrrolidin-3-yl)-1H-imidazole-2-carboxylate
1-(2-chloro-6-methylphenyl)-3-(2-hydroxyethyl)-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
2-(3-chlorophenyl)-2-hydroxy-N-methyl-N-[(3-methylpyridin-4-yl)methyl]acetamide
5-(8-methoxy-2H-chromen-3-yl)-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-(1-ethynylcyclohexyl)-1-(2-methoxyethyl)pyrrolidine-3-carboxamide
N-(4-fluorophenyl)-1-(3-methylbenzoyl)piperidin-3-amine
4-butyl-11-{[(4-methoxyphenyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2-(3,4-dichlorophenyl)morpholine
7-cyclopentyl-2-{2-methylthieno[2,3-d]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decan-6-one
2-(1-{1,9-dioxaspiro[5.5]undecan-4-yl}azetidin-3-yl)pyridine
N,N-dimethyl-2-{[2-(morpholin-4-yl)butanamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-(2-methoxyphenyl)-3-{1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-(2-ethoxyethyl)-5-[3-(morpholin-4-yl)azetidine-1-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-cyclopropyl-1-[1-(2-methylquinolin-4-yl)piperidin-4-yl]piperidine-3-carboxamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(pyridin-2-ylsulfanyl)acetamide
{1-[(6-methylpyridin-2-yl)methyl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
2-(2,3-dihydro-1H-isoindole-2-carbonyl)-8-fluoroquinoline
(1R,5R)-6-(2-methoxyethyl)-3-[4-(trifluoromethyl)pyridin-2-yl]-3,6-diazabicyclo[3.2.2]nonane
3-[({1-[3-(trifluoromethyl)benzoyl]piperidin-3-yl}oxy)methyl]pyridine
3-(2H-1,3-benzodioxol-5-yl)-5-(4,4,4-trifluorobutyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-(4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-oxobutan-2-yl)acetamide
4-hydroxy-1-(2-methyl-5-propylpyrimidin-4-yl)piperidine-4-carboxylic acid
3-cyclopropyl-5-[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazole
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1,3-thiazol-2-ylmethyl)pyrrolidin-3-yl]-5-methyl-1,2-oxazole-3-carboxamide