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N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
2-{[5-(3-chloro-5-fluoro-4-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}pyridine
ethyl 3-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]pyrrolidine-1-carboxylate
1-(4-benzylpiperazine-1-carbonyl)-6-(naphthalen-1-ylmethyl)-6-azaspiro[2.5]octane
2-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
5-[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]pyridine-2-carbonitrile
2-{4-[(3,4-difluorophenyl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
(2R)-2-methoxy-2-phenyl-1-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
benzyl (1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
1-[4-(hydroxymethyl)piperidin-1-yl]-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
1-[4-(aminomethyl)benzoyl]-4-(1H-imidazol-4-ylmethyl)-1,4-diazepan-6-ol
N-{[5,8-dimethoxy-2-(4-methylphenyl)quinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(dimethylamino)ethyl]propanamide
2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
2-{[2-(azepan-1-yl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-ethyl-N-(2-methylprop-2-en-1-yl)acetamide
ethyl 1-(but-2-ynoyl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
4-({1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-2-yl}methyl)morpholine
ethyl 1-{2-[1-cyclopentyl-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperidine-2-carboxylate
9-(5-fluoro-2-methylbenzoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,2,4-trimethylbenzamide
4-(1H-imidazol-1-yl)-1-[2-(2-oxopyrrolidin-1-yl)propanoyl]piperidine-4-carboxylic acid
3-methyl-7-(2-phenoxybenzoyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-(2-hydroxyethyl)-N-(thiophen-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-[2-(3-methoxyphenyl)ethyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-(2-{1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
3-(furan-3-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
methyl 1-benzyl-5-[(2-methylpropyl)amino]-3-(oxolane-2-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
N-[(3,4-dimethoxyphenyl)methyl]-2-(methoxymethyl)-6-methyl-1-(naphthalen-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
3-(3-fluorophenyl)-4-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}-1H-pyrazole
2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
2-cyclohexyl-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-benzoxazole-6-carboxamide
1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
3-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-(2-hydroxypyridin-3-yl)urea
4-{1-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]piperidin-3-yl}benzoic acid
2-{4-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]piperazin-1-yl}ethan-1-ol
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylbenzamide
N-[(3-tert-butyl-1,2,4-oxadiazol-5-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-[(4-fluorophenyl)methyl]-N-{2-[2-(trifluoromethyl)phenyl]ethyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
7-[(2-fluorophenyl)methyl]-2-(pyridin-2-ylmethyl)-2,7-diazaspiro[4.5]decane
ethyl 1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(pyridin-3-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
2-methoxy-6-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenol
ethyl 4-({3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-ethyl-1-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N,4,6-trimethylpyrimidin-2-amine