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1-(methoxymethyl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}cyclobutane-1-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-[(1-methyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(3aR,6aR)-2-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2-hydroxyphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
7-[(3,4-difluorophenyl)methyl]-2-(2-methoxypyrimidine-5-carbonyl)-2,7-diazaspiro[4.5]decane
1-methyl-3-(3-phenyl-1,2,4-thiadiazol-5-yl)-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)urea
8-(4-aminopyrimidin-2-yl)-2-cyclopentyl-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(2-phenylethyl)piperidin-3-yl]furan-3-carboxamide
1-{3-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl}ethan-1-one
3-{[(2-methyl-5-propylpyrimidin-4-yl)amino]methyl}-1λ6-thiolane-1,1-dione
5-chloro-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1,3-dimethyl-1H-pyrazole-4-sulfonamide
(3R,5S)-5-{3-[(2-methoxyphenyl)methyl]-1-[(4-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}pyrrolidin-3-ol
5-{4-phenyl-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}pentan-1-amine
4-(2,4-dioxoimidazolidin-1-yl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}benzamide
1-cyclopentyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
2-cyclopentyl-1-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
8-(2-amino-2-methylpropyl)-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(4-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}morpholin-3-yl)methanol
8-[(2,3-difluorophenyl)methyl]-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-(cyclopropylmethyl)-1-methyl-4-(1,3-thiazol-2-ylmethyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{3-[(5-methylpyridin-2-yl)amino]propyl}-4-sulfamoylbenzamide
1-(3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl)-4-(4-methoxyphenyl)butane-1,4-dione
(3R,4S)-1-(2-methoxy-4-methylbenzoyl)-4-propylpyrrolidin-3-amine
N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-1-(piperidin-1-yl)ethan-1-one
2-{4-[4-(3-methylbutyl)-2,5-dioxoimidazolidin-4-yl]piperidin-1-yl}pyridine-3-carboxylic acid
(1R,3S,5S)-8-(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)-8-azabicyclo[3.2.1]octan-3-ol
5-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)pentan-1-ol
8-methoxy-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-amine
1-{3,9-diazaspiro[5.5]undecan-3-yl}-3-(4-hydroxyphenyl)propan-1-one
2,6-dimethyl-7-[1-(oxan-4-yl)-4-phenyl-1H-imidazol-5-yl]heptan-2-ol
1-[1-(1-ethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(2-chlorophenyl)methyl]-N-cyclohexyl-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-(1,3-benzoxazol-2-ylmethyl)-N-methyl-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
N-methyl-1-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]-N-(pyridin-3-ylmethyl)piperidin-4-amine
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(2-methoxyphenoxy)-2-methylpropanamide
(1R,5R)-3-(4-chloro-3-methyl-1H-pyrazole-5-carbonyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-(2,2-dimethyloxane-4-carbonyl)-1-(2-methoxyphenyl)-2,2-dimethylpiperazine
1-[4-(4-{[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
(1S,5R)-6-(cyclopropylmethyl)-3-[(3-ethoxy-4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-[3-(1-methylpiperidin-2-yl)propanoyl]-4-phenylpiperidine-4-carbonitrile
(3R,4S)-4-cyclopropyl-1-[4-(morpholine-4-carbonyl)benzoyl]pyrrolidin-3-amine
(3S,4R)-3-benzyl-1-(3,4-dimethylbenzoyl)-4-methylpiperidin-4-ol
2-[4-(1-cyano-1-methylethyl)phenyl]-2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}acetic acid
N-(1-hydroxybutan-2-yl)-2-(morpholin-4-yl)-N-(thiophen-3-ylmethyl)benzamide
({1-[(1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)(methyl)amine
1-cyclohexyl-4-[(2S)-5-oxopyrrolidine-2-carbonyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one