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5-{1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1H-1,2,3-triazol-4-yl}-2-(propan-2-yl)pyrimidine
N-[(8-methoxyquinolin-5-yl)methyl]-N,3,4,7-tetramethyl-1H-indole-2-carboxamide
2-[(2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}phenyl)formamido]acetamide
5-chloro-2-[(3S)-3-ethylmorpholine-4-carbonyl]-3-phenyl-1H-indole
(3aR,6aR)-2-acetyl-5-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[4-(3-propoxypiperidin-1-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl]pyridine
7-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(2-methoxyethyl)-N-(2,2,2-trifluoroethyl)-1,3-benzoxazole-6-carboxamide
2-[2-oxo-4-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)piperazin-1-yl]benzonitrile
1-[2-(2-oxopyrrolidin-1-yl)acetyl]-4-phenoxypiperidine-4-carboxylic acid
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-4-(thiophen-2-yl)butan-1-one
3-(hydroxymethyl)-1-{[4-(morpholine-4-sulfonyl)phenyl]methyl}piperidin-3-ol
1-acetyl-N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]piperidine-3-carboxamide
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-4-(piperidin-1-yl)butanamide
1-cyclopropyl-3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
N-[3-(1H-imidazol-1-yl)propyl]-2-methyl-N-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrimidine-3-carboxamide
ethyl 4-[(3-fluorophenyl)methyl]-1-(1H-pyrazol-3-ylmethyl)piperidine-4-carboxylate
3-(4-fluorophenyl)-4-[5-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-1H-pyrazole
5-cyclopropanecarbonyl-1'-(4-methoxybenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 3-acetamido-1-(3-methylbutyl)-5-[(1,2,3,4-tetrahydronaphthalen-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]methylamine
4,6-dimethyl-2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
1-hexyl-4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidine
3-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}-6-(propan-2-yl)pyridazine
5-benzyl-1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
4-methoxy-3-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]benzene-1-sulfonamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-methyl-1-benzofuran-5-carboxamide
N-[2-(dimethylamino)ethyl]-2-(4-hydroxyphenyl)-N-[(3-methylthiophen-2-yl)methyl]acetamide
N-{[3-(methylsulfanyl)phenyl]methyl}-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(furan-2-ylmethyl)methylamine
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-2-(1H-pyrazol-1-yl)benzamide
2-{[(1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)oxy]methyl}pyridine
5-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}-2-(pyrrolidin-1-yl)-1,3-thiazole
3-butanamido-N-[(1-propylpiperidin-3-yl)methyl]benzamide
(1R,5R)-6-[2-(benzyloxy)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
6-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}quinoxaline
N-(1-methyl-1H-1,2,4-triazol-3-yl)-3-{[3-(2-methylpropyl)morpholin-4-yl]methyl}benzamide
methyl 3-(5-methoxyfuran-2-carbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(7-benzoyl-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]thiophene-2-sulfonamide
1-[(3,5-dimethylphenyl)methyl]-4-(2,3,6-trifluorobenzoyl)piperazin-2-one
(1R,3S,5S)-8-[2-(1H-indol-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-8-azabicyclo[3.2.1]octan-3-ol
2,6-difluoro-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)benzamide
3-cyclopentyl-5-(2,5-dimethoxyphenyl)-1H-1,2,4-triazole
6-chloro-3-({[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]amino}methyl)-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
4-chloro-2-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methyl-1H-indole
N-[1-(4-{4-[(4-fluorophenyl)sulfanyl]piperidine-1-carbonyl}phenyl)-1H-pyrazol-4-yl]acetamide
6-methyl-5-{5-[(propan-2-yloxy)methyl]-1,2,4-oxadiazol-3-yl}-N-propyl-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
methyl 4-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
3-(azocan-1-yl)-1-(4-ethylpiperazin-1-yl)propan-1-one