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methyl({[5-(oxolan-2-yl)thiophen-2-yl]methyl}){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-cyclopropanecarbonyl-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}piperidine-4-carboxamide
11-{[(2,3-difluorophenyl)methyl]amino}-4-[2-(1H-indol-3-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-(butan-2-yl)-5-methyl-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-{[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
7-(2-methoxyethyl)-2-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(thian-4-yl)piperazin-2-yl}ethan-1-ol
N-[1-(pyrazin-2-yl)piperidin-3-yl]imidazo[1,2-a]pyridine-6-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-1-{4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-carboxamide
2-methyl-4-(3-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}phenyl)butan-2-ol
N-[3-(4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}piperidin-1-yl)phenyl]-3-(trifluoromethyl)benzamide
N-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-1,3-dimethyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
6-[2-(naphthalen-2-yl)acetyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(2-methylprop-2-en-1-yl)benzamide
2-[4-(1H-indol-2-ylmethyl)-1-[(4-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-(dimethylamino)-1-(4-hydroxypiperidin-1-yl)-2-(4-methylphenyl)ethan-1-one
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
5-(furan-2-yl)-3-({2-[5-(oxan-2-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole
2-methyl-N-{4-[4-(pyrrolidin-1-yl)piperidine-1-carbonyl]phenyl}furan-3-carboxamide
1-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-3-[5-(2-methylphenyl)-1,3,4-thiadiazol-2-yl]urea
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(oxan-4-yl)acetamide
N-[(3R,4R)-3-hydroxy-1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl]pyrazine-2-carboxamide
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-[1'-(3,4-dimethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
2-methyl-6-{1-[1-(propan-2-yl)piperidine-4-carbonyl]piperidin-3-yl}pyrimidin-4-ol
[1-(4-aminopyrimidin-2-yl)-4-[(2-chlorophenyl)methyl]piperidin-4-yl]methanol
N-({7-[2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)propane-1-sulfonamide
2,3-dimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-indole-7-carboxamide
4-methoxy-2-[({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}amino)methyl]phenol
(4S)-3-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
3-methyl-2-({4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
1-(4-{[(6-methylpyridin-2-yl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
4-(2,6-dimethylquinoline-3-carbonyl)-3-(3-fluorophenyl)piperazin-2-one
5-[(3-methoxyphenyl)methyl]-3-methyl-5-[1-(pyridin-3-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
N-(dicyclopropylmethyl)-N-methyl-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
(2S,4S)-N-ethyl-1-(oxan-4-yl)-4-[3-(pyridin-4-yl)propanamido]pyrrolidine-2-carboxamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-3,4,5-trimethoxy-N-(pyridin-4-ylmethyl)benzamide
8-[(3,5-dimethylphenyl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N4-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
methyl({[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})(quinolin-5-ylmethyl)amine
N-[2-(diethylamino)ethyl]-1,3,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
9-methoxy-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-2-(4-methyl-2-oxo-1,2-dihydroquinolin-1-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4-(morpholin-4-yl)butan-1-one
1-(4-ethoxy-2-fluorophenyl)-3-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]urea
1-methyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[1-benzyl-5-(ethoxymethyl)-1H-1,2,4-triazol-3-yl]acetamide