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N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
3-(1,2-oxazinan-2-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]propanamide
1-[1-(5-fluoropyrimidin-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N,1-dimethyl-N-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}pyrrolidin-3-amine
1-methyl-3-(propan-2-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
(3aS,6aS)-2-(oxan-4-yl)-5-(pyrimidin-5-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(furan-3-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
4-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyloxan-4-amine
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N-(2-fluoroethyl)-3-{[1-(1,3-thiazol-2-yl)propyl]sulfamoyl}benzamide
(1R,2S,4R)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
N-[2-(dimethylamino)ethyl]-N-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}oxolane-2-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,6,6-trimethyl-5-oxothiomorpholine-3-carboxamide
methyl 8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-(3-methoxyphenyl)-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]azetidine
1-{4-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]phenyl}pyrrolidin-2-one
2-{2-[2-(4-ethylpiperazin-1-yl)ethoxy]phenyl}-6-methyl-1H-1,3-benzodiazole
5-(4-fluorophenyl)-2-methyl-4-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}pyrimidine
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]piperidin-4-amine
N-methyl-1-[(2-methylphenyl)methyl]-N-(pyridin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
5-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]pyrazin-2-ol
3-[({[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(3-chloro-5-methoxybenzoyl)-4-(hydroxymethyl)piperidin-4-ol
7-{3-[(4-fluorophenyl)formamido]propanoyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-5-oxopyrrolidine-3-carboxylic acid
1-{[4-methoxy-3-(prop-2-en-1-yl)phenyl]methyl}-2-methyl-1,4-diazepan-5-one
4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
(4aS,7aR)-1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-[(4-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
1-[2-(morpholin-4-yl)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
7-cyclopentyl-2-(4-fluorobenzenesulfonyl)-2,7-diazaspiro[4.5]decan-6-one
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)acetamide
ethyl 2-{[2-(azocane-1-carbonyl)phenyl]amino}acetate
1-{1-[2-(propylamino)benzoyl]piperidin-4-yl}pyrrolidin-2-one
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl})amine
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(5-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
N-(1-hydroxybutan-2-yl)-2-(methylamino)-N-(thiophen-2-ylmethyl)pyridine-3-carboxamide
3-[(2-hydroxyethyl)({[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl})amino]-1λ6-thiolane-1,1-dione
2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
4-({[2-(dimethylamino)ethyl][(2-methylphenyl)methyl]amino}methyl)benzoic acid
1-[(4-fluorophenyl)methyl]-4-{[6-methyl-4-(thiomorpholin-4-yl)quinazolin-2-yl]methyl}piperazin-2-one
3-hydroxy-1-(2-phenylethyl)-3-{[(pyrimidin-4-ylmethyl)amino]methyl}piperidin-2-one
6-methyl-N-(1-methylpiperidin-4-yl)-4-oxo-N-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-[3-(2-chlorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[3-(morpholin-4-yl)propyl]acetamide
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl){[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
1-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-3-yl]-2-phenylethan-1-one
5-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-1-cyclopropylpiperidin-2-one
(3R)-1-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}pyrrolidin-3-ol
N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[4-(morpholin-4-yl)butyl]acetamide