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1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[(3-methoxyphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
2-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]pyridine-4-carboxylic acid
5-(2-{2-[(1,3-benzothiazol-2-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
3-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-5-(3-methoxyphenoxymethyl)-1,2-oxazole
(3S,4R)-3-methoxy-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)benzoyl]piperidin-4-amine
2-ethyl-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
N-{3-[(5-cyclobutyl-1,3,4-oxadiazol-2-yl)amino]propyl}-4-methylbenzene-1-sulfonamide
N-cyclopentyl-N-(3-phenylprop-2-yn-1-yl)-2-(pyridin-3-yloxy)acetamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)furan-3-carboxamide
3-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1H-pyrazol-5-amine
2-[4-(quinolin-6-yl)phenoxy]propanamide
1-(dimethyl-1,3-thiazole-4-carbonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperazine
2-ethyl-N-(3-ethylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-{[4-(2-fluorophenoxy)piperidin-1-yl]methyl}-3-hydroxy-1-methylpiperidin-2-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-[3-({methyl[1-(pyridin-2-yl)propyl]amino}methyl)phenoxy]acetamide
2-(2-{[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]amino}ethyl)-6-methyl-3,4-dihydropyrimidin-4-one
1-cyclopentanecarbonyl-4-(2-phenylazetidine-1-carbonyl)piperidine
2-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]quinazolin-2-yl}ethan-1-amine
2-(3-chloro-5-fluoro-4-methoxyphenyl)-1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-1H-imidazole
9-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
9-methoxy-4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-yl]methyl})amino]ethan-1-ol
4-(2,8-dimethylquinoline-4-carbonyl)-1-methylpiperazine-2-carboxylic acid
8-(2-hydroxypropyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}[(4-ethylphenyl)methyl]methylamine
3,5-dimethyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,2-oxazole-4-sulfonamide
1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
1-(4-{[(cyclohexylmethyl)amino]methyl}-2-methoxyphenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
4-[(benzyloxy)methyl]-7-hydroxy-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
1-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}urea
4-[(2,4-dimethoxyphenyl)methyl]-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
N-[2-(3-methoxyphenyl)-1-[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
5-cyclopropyl-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1,3-oxazole-4-carboxamide
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
4-chloro-3-(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carbonyl)-1H-pyrazol-5-amine
2-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]pyridine-3-carboxamide
3-{[1-benzyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
2-{[4-(2-methylphenyl)-5-[(propan-2-yloxy)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-{[2-(2-fluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}-4-methoxyphenol
1-{[4-(2-aminoethyl)phenyl]methyl}-4-(oxan-4-yl)-1,4-diazepan-6-ol
2-(2,3-dimethoxyphenyl)-1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]ethan-1-one
3-(6-fluoropyridin-3-yl)-1-{[1-(pyridin-2-yl)piperidin-3-yl]methyl}urea
5-{[(4aS,7aR)-4-(2-methoxyacetyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
1-[(2-fluorophenyl)methoxy]-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,8-diazaspiro[4.5]decan-2-one
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[3-(1H-pyrazol-1-yl)propyl]amine
6-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
3-fluoro-N-(1-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-(2-chlorophenyl)-1-methyl-3-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]pyrrolidine-2,5-dione