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(1S,5R)-3-(5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[(2-methoxyethyl)amino]-5-methyl-N-[3-(pyridin-4-yl)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
methyl 4-[(4aR,8aS)-6-(1H-indole-2-carbonyl)-decahydro-1,6-naphthyridine-1-carbonyl]benzoate
1-(2-cycloheptyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
3-{5-[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}pyridazine
[(2,4-dimethoxy-3-methylphenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
5-(3,4-dimethoxyphenyl)-N-[2-(1H-imidazol-1-yl)ethyl]-1,2,4-triazin-3-amine
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methylpropanamide
(3S,4R)-1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-phenylpyrrolidine-3-carboxylic acid
(1R,5R)-6-benzyl-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
3-[1-(4-chloro-1H-pyrrol-2-yl)-N-(2-phenylethyl)formamido]propanamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(2,2-dimethyloxan-4-yl)-5-methoxybenzamide
methyl(pyridin-3-ylmethyl)[2-(pyrimidin-2-yloxy)hex-5-en-1-yl]amine
5-{[2-(diethylamino)ethyl](methyl)amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-[2-(pyridin-3-yloxy)ethyl]piperidine-3-carboxamide
(1R,3S)-7-[(1-benzyl-1H-indol-6-yl)methyl]-7-azaspiro[3.5]nonane-1,3-diol
2-{1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
2,6-dimethoxy-N-{[6-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
2-[3-(1H-imidazol-1-yl)propyl]-9-(pyridine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[7-(1-benzofuran-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-(3-fluorophenyl)acetamide
N-[2-(3-methylthiophen-2-yl)ethyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
[(1-ethylpiperidin-3-yl)methyl](methyl)[(3-methyl-1H-indol-2-yl)methyl]amine
methyl 3-({[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]carbamoyl}amino)-4-methoxybenzoate
3-[1-(1-benzothiophen-2-ylmethyl)piperidin-3-yl]-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N,1-dimethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2-propyl-1,3-thiazole-4-carboxamide
N-[(4-fluorophenyl)methyl]-N-methyl-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
6-ethyl-1,5-dimethyl-2-oxo-N-[(1R,2S)-2-phenylcyclopropyl]-1,2-dihydropyridine-3-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]propanamide
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]ethan-1-one
4-methyl-1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}pentan-1-one
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)benzamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
4-[4-(3-cyclohexylpropanoyl)piperazin-1-yl]-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
7-(9H-fluoren-2-ylmethyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-{2-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-2-oxoethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
9-(6-methylpyrimidin-4-yl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]propanamide
2-(2-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}phenoxy)propanoic acid
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-amino-4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-6-(3-methylphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-3-[2-(ethylsulfanyl)ethyl]urea
7-(2-methoxyacetamido)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-N-[(2-ethoxyphenyl)methyl]-N-ethylpropanamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5,6-dimethylpyrimidin-4-amine
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(pent-2-yn-1-yl)piperidine
2-(dimethylamino)-N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]benzamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[3-(5-methylthiophen-2-yl)-1H-pyrazol-1-yl]acetamide