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1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(oxolan-2-ylmethyl)-4-phenyl-1H-imidazole
5-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)-2,1,3-benzothiadiazole
N-({8-[(2-chloro-6-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-3-fluorobenzamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N-(3,4-dimethoxyphenyl)-1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-3-amine
2-butyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
2-(4-{[3-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}phenoxy)ethan-1-ol
2-[2-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
ethyl 2-(2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methylacetamido)acetate
3-({1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}amino)azepan-2-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(1-methylcyclopropanecarbonyl)pyrrolidin-3-yl]methanol
3-[1-(pyridin-2-yl)piperidin-4-yl]propanamide
1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]urea
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[4-(hydroxymethyl)piperidin-1-yl]methyl}piperidin-2-one
[(3-{2-[4-(2H-1,3-benzodioxole-5-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(1,3-thiazol-4-ylmethyl)amine
4-(1H-imidazol-1-ylmethyl)-1-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-ol
2-(4-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-yl)pyridine
N-cyclopropyl-4-({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}amino)pyridine-2-carboxamide
4-chloro-2-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}phenol
1-[1-(but-2-ynoyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-4-carboxamide
N-[1-({[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
2-[4-(6,8-dimethylquinolin-4-yl)-1-methylpiperazin-2-yl]ethan-1-ol
methyl 4-{[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}butanoate
(3S,4R)-4-(hydroxymethyl)-1-(4-phenyl-1H-imidazole-5-carbonyl)piperidin-3-ol
3-(3-fluorophenyl)-4-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-pyrazole
methyl (3aS,6aS)-2-(3-methylfuran-2-carbonyl)-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylate
4-(2-{2-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}ethyl)morpholine
6-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
2-(4-fluorophenyl)-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)acetamide
N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
(4aS,8aS)-2-(2,5-dimethylbenzenesulfonyl)-decahydro-2,7-naphthyridin-4a-ol
3,4-dimethoxy-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-{[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazol-3-yl]acetamide
(3S,4R)-4-(hydroxymethyl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-3-ol
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-2-(pyrrolidin-1-yl)-6-(thiophen-3-yl)pyridine-3-carboxamide
(4aS,7aR)-N-(3-fluorophenyl)-4-(1H-imidazol-4-ylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-[1-(4-methoxyphenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]propanamide
1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
3-acetamido-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)benzamide
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-methyl-2-phenyl-N-(thian-4-yl)acetamide
{2-[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]phenyl}methanol
5-chloro-N-(2-hydroxypropyl)-15-methyl-13-oxo-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
2-(butylsulfanyl)-6-(3-methoxypyrrolidin-1-yl)pyrimidin-4-amine
1-(1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
methyl 1-(benzyloxy)-8-(2-methylpropyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-{2-[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidine-1-carbonyl]phenyl}ethan-1-one
N-{1-[(5-cyclopentylthiophen-2-yl)methyl]pyrrolidin-3-yl}acetamide
1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)but-3-en-1-one
1-[3-({[(3-chlorophenyl)methyl]amino}methyl)phenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol