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5-(3-fluorophenoxymethyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
2-(4-{[(3-cyano-4-ethoxyphenyl)carbamoyl]amino}piperidin-1-yl)-N-cyclopropylacetamide
1-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
3-(2-chlorophenyl)-1-cyclopentyl-3-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}pyrrolidine-2,5-dione
9-[6-(4-fluorophenyl)pyridazin-3-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-[1-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)pyrrolidin-2-yl]-1,3-thiazole
2-{1-[(4-ethoxyphenyl)methyl]-4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
2-ethyl-4-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}morpholine
N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyridine-2-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(pyridin-3-ylmethyl)benzamide
1-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-2-(1-propylpiperidin-4-yl)ethan-1-one
3-(4-methyl-1,3-thiazol-5-yl)-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
4-(benzenesulfonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{[7-(2,5-difluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
2-{1-cyclohexyl-5-[(3-phenylpyrrolidin-1-yl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
1-(3-{[7-acetyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
1-{2-oxo-1-[2-(piperidin-1-yl)ethyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-6-yl}-4-phenylbutane-1,2-dione
3-(3-hydroxy-3-methylbutyl)-N-[3-(3-oxopiperazin-1-yl)propyl]benzamide
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
5-{[2-(2-fluorophenyl)ethyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(4aS,7aR)-1-[2-(1H-imidazol-2-yl)benzoyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6,7-dimethoxy-2-(1-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
2-[1-ethyl-2,4-dioxo-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
1-(2H-1,3-benzodioxol-5-yl)-3-[2-(methylsulfanyl)ethyl]-5-(oxan-2-yl)-1H-1,2,4-triazole
3-(3-methylthiophene-2-carbonyl)-1-[4-(trifluoromethyl)benzenesulfonyl]piperidine
3-{2-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
N-[(7-chloro-4-{[(4-fluorophenyl)methyl]amino}quinazolin-2-yl)methyl]cyclohex-3-ene-1-carboxamide
5-methyl-2-(3-methyl-3-phenylpiperidine-1-carbonyl)pyridine
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(3-ethynylbenzoyl)-N-methylpiperidin-3-amine
2-(4,6-dimethylpyrimidin-2-yl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-fluoro-1-methyl-2-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)-1H-indole
8-[(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
6-(benzyloxy)-1-cyclohexyl-4-(5-methylpyrazine-2-carbonyl)-1,4-diazepan-2-one
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-(pyridin-4-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-methyl-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-N-(propan-2-yl)piperidine-4-carboxamide
5-{1-[(4-methoxynaphthalen-1-yl)methyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
9-(5-methoxyfuran-2-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-(4-{[4-(3-fluorophenoxy)piperidin-1-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
N3-(cyclohexylmethyl)-1-cyclopropyl-N5-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(4-fluorophenyl)methyl]-2-(4-hydroxypiperidin-1-yl)-6-[4-(methylsulfanyl)phenyl]pyridine-3-carboxamide
3-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
1-(2-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-1-methylurea
1-(2-{methyl[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidine
(4aS,7aR)-1-(3-acetylbenzoyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aS,7aR)-1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-phenyl-5-[1-(3-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazole
{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
methyl 4-{[(2-{5-oxo-1-[2-(propan-2-yloxy)ethyl]pyrrolidin-2-yl}ethyl)amino]methyl}benzoate