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1-{5-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-(3-methoxybenzoyl)piperazine
N-[(7-{[4-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-4-[3-(trifluoromethyl)benzoyl]-1,4-diazepan-2-one
2-ethyl-8-(2-methylpyridin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
2-(3-methoxypropyl)-8-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-[4-(1-benzothiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-1-(dimethylamino)propan-2-ol
N-({7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
3-hydroxy-1-methyl-3-{[(1-phenylcyclopropyl)amino]methyl}piperidin-2-one
4-(3,4-difluorobenzoyl)-6-methoxy-1-[(4-methoxyphenyl)methyl]-1,4-diazepan-2-one
N-(adamantan-1-ylmethyl)-2-[3-(2-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
4-(2-fluoro-5-methylphenoxy)-1-(pyrrolidine-1-carbonyl)piperidine-4-carboxylic acid
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(3-methoxypropyl)-N-methyl-1,3-oxazole-4-carboxamide
(5-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}furan-2-yl)methanol
2-(2-methoxyethyl)-8-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(3,5-dimethoxyphenyl)-3-{1-[2-(methylsulfanyl)acetyl]piperidin-3-yl}propanamide
2-{4-[(2-methoxyphenyl)methyl]-1,4-diazepan-1-yl}-4,6,7-trimethylquinazoline
7-methoxy-3-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
ethyl 1-benzyl-5-[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
6-ethyl-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-methylquinoline-4-carboxamide
2-(3-phenylpropyl)-8-(pyrrolidine-1-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-[2-(2-chlorophenyl)ethyl]-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-N,N-dimethylacetamide
1-{2-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]phenyl}-1,3-diazinane-2,4-dione
1-{[4-hydroxy-1-(1-phenylpiperidin-4-yl)azepan-4-yl]methyl}-3,3-dimethylurea
(1S,5R)-3-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 1-{2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperidine-2-carboxylate
3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-(3,4-dimethylphenyl)piperidine-1-carboxamide
2-[1-(2-chlorophenyl)-5-(oxolan-3-yl)-1H-1,2,4-triazol-3-yl]acetamide
4-benzyl-1-(pent-2-yn-1-yl)-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]-3-[(thiophen-2-ylmethyl)amino]benzamide
1-[(2,6-difluorophenyl)methyl]-5-(2-{[(3-methylphenyl)methyl]amino}ethyl)pyrrolidin-2-one
5-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
5-methyl-4-(4-methylpiperazin-1-yl)-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,2,5-thiadiazole-3-carboxamide
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pent-4-enamide
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-2-(pyridin-2-ylsulfanyl)acetamide
(2R,6R)-4-[(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)methyl]-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(3-{2-[1-(3-chloropyridin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
4-(6-chloro-1,3-benzothiazol-2-yl)-1,4-oxazepan-6-ol
1-[(2-chlorophenyl)methyl]-N-cyclohexyl-N-(prop-2-yn-1-yl)-1H-1,2,3-triazole-4-carboxamide
N-benzyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[3-(morpholine-4-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(thiophen-2-yl)ethan-1-one
2-(3-{[3-(piperidin-1-yl)pyrrolidin-1-yl]methyl}phenoxymethyl)pyridine
1-(2-ethylphenyl)-3-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}urea
1-(2-methoxyethyl)-3-(2-phenylethyl)-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}pyrrolidin-3-yl)methyl]benzoic acid
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(3-fluoropyridine-2-carbonyl)pyrrolidine-3-carboxylic acid
N-[(4-methanesulfonylmorpholin-2-yl)methyl]cyclopentanamine