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3-chloro-4-{[1-(cyclopropylmethyl)piperidin-4-yl]oxy}-N-[2-(dimethylamino)ethyl]benzamide
(1S,5R)-3-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-phenyl-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-4-yl)ethan-1-one
1-cyclohexyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}piperidine-4-carboxamide
2-{2-methyl-4-[(4-methylphenyl)methyl]-3-oxopiperazine-1-carbonyl}benzonitrile
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
(3aS,6aS)-5-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-N,N-dimethyl-octahydropyrrolo[3,4-b]pyrrole-1-carboxamide
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]acetamide
N,N-dimethyl-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}pyrrolidin-3-amine
4-amino-N-(cyclohex-1-en-1-ylmethyl)pyridine-2-carboxamide
5-methoxy-1,3-dimethyl-6-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
8-(3-{[(4-fluorophenyl)methyl]sulfanyl}propanoyl)-2,8-diazaspiro[4.5]decan-3-one
5-(3-phenylpropyl)-5-[1-(quinolin-7-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
3-[2-(3-acetylpiperidin-1-yl)-2-oxoethyl]-1-cyclopentyl-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
1-[(2,5-dimethylphenyl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
5-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-[3-(morpholin-4-yl)propyl]-1,2-oxazole-3-carboxamide
methyl 4-[(4-cyclohexyl-6-hydroxy-3-oxo-1,4-diazepan-1-yl)methyl]benzoate
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-N-methyl-4-oxo-N-(pyridin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-(3-fluorophenyl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-{3-cyclobutyl-6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-1H-pyrazole-3-carboxylic acid
3-[(benzylsulfamoyl)amino]-N-(1,3-thiazol-2-yl)propanamide
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(piperidin-1-yl)ethyl]amine
2-amino-6-(4-hydroxy-2-methylphenyl)-4-[2-(propylamino)pyrimidin-5-yl]pyridine-3-carbonitrile
N4-(1H-imidazol-2-ylmethyl)-7-[(2R)-oxolane-2-carbonyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-({7-[(3,5-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenoxyacetamide
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol
3-(4-methoxyphenyl)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
7-[2-(4-oxo-3,4-dihydro-1,2,3-benzotriazin-3-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-(3-chloro-5-fluoro-4-methoxyphenyl)-1-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-imidazole
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
methyl 6-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-2-[(2-methoxyethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
ethyl 4-[1-(cyclopropylmethyl)-3-[(1,3-thiazol-2-ylmethyl)carbamoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]piperidine-1-carboxylate
2-methyl-4-(4-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}phenyl)butan-2-ol
4-ethyl-6-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-N,N-dimethylpyrimidin-2-amine
2-amino-6-(6-methoxypyridin-3-yl)-4-[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
9-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2-fluorophenyl)-3-(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-3-yl)propanamide
3-amino-1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}pyrrolidine-3-carboxylic acid
N-(2,3-dihydroxypropyl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
N-[3-(azepan-1-yl)propyl]-N,1-dimethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
methyl 5-[2-(3-chloro-4-hydroxyphenyl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-[(1R,2S)-2-phenylcyclopropyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
(3S)-1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)pyrrolidin-3-amine
N-[(3R,4R)-3-hydroxy-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl]pyridine-3-carboxamide
1-[(5-propylfuran-2-yl)methyl]-4-(thiophen-2-ylmethyl)piperazine
N-cyclopentyl-5-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide