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N-(1H-imidazol-2-ylmethyl)-N-methylquinoxaline-5-carboxamide
1-benzyl-5-acetamido-N,2-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
4-[3-(morpholin-4-yl)phenoxy]oxane-4-carboxylic acid
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(1H-pyrazol-1-yl)benzamide
2-{1-[(3,4-difluorophenyl)methyl]-4-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
(5S,9aS,9bS)-2-[(2-methylphenyl)methyl]-5-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-5-methylthiophene-2-carboxamide
2-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-6-methylpyridine
methyl (2S,4R)-4-(4-methylbenzamido)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxylate
ethyl 3-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carbonyl]amino}propanoate
ethyl 1-[2-(cyclopentylmethyl)-6-methyl-4-oxo-1-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carbonyl]piperidine-2-carboxylate
1-(4-{[(2R)-hexan-2-yl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-cyclohexyl-N-methyl-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-(furan-3-ylmethyl)-1-methyl-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
4-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)morpholine
3-(but-2-yn-1-yl)-5-{1-[2-(3-fluorophenyl)acetyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,8-dimethylquinoline
5-ethyl-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-1H-pyrrole-2-carboxamide
3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
4-methyl-2-(propan-2-yl)-6-{4-[3-(propoxymethyl)pyrrolidin-1-yl]piperidin-1-yl}pyrimidine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
5-(2-methylpropyl)-1-(pentan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
ethyl 4-(3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)piperazine-1-carboxylate
N-methyl-2-[2-(morpholin-4-ylmethyl)-4-(pyrazin-2-yl)phenoxy]-N-[2-(pyridin-2-yl)ethyl]acetamide
4,4,4-trifluoro-1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butan-1-one
(3R,5R)-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
1-(4-{4-[(2,2-diphenylethyl)amino]piperidin-1-yl}benzoyl)piperidin-3-ol
1-{2-hydroxy-3-[4-methoxy-2-({[2-(3-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
3-{[methyl(propyl)carbamoyl]methyl}-N-[3-(methylsulfanyl)phenyl]morpholine-4-carboxamide
4-[5-(3,5-dimethoxyphenoxymethyl)-1,2,4-oxadiazol-3-yl]benzoic acid
4-{[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
2-ethyl-7-{[(3S)-3-ethylmorpholin-4-yl]methyl}-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
(1S,5R)-6-(cyclobutylmethyl)-3-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[(4-fluorophenyl)methyl]-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-1,4-diazepan-2-one
3-(3-methoxyphenyl)-N-{[8-(pyridin-4-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
5-ethyl-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1,3-oxazole-4-carboxamide
(1R,5S)-6-[(2-cyclohexylpyrimidin-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-methyl-1-propyl-N-(2,2,2-trifluoroethyl)-1H-pyrazole-4-carboxamide
5-chloro-N-[(2-methoxyphenyl)methyl]-4,6-dimethyl-2-oxo-N-propyl-1,2-dihydropyridine-3-carboxamide
methyl 3-(2-methoxyacetyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-2-(1H-indazol-3-yl)acetamide
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
N4-[1-(4-methanesulfonylphenyl)ethyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
3-(3-fluorophenyl)-1-methyl-3-(2-oxo-2-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}ethyl)pyrrolidine-2,5-dione
1-methyl-2-oxo-N-[3-(3-oxopiperazin-1-yl)propyl]-1,2-dihydroquinoline-4-carboxamide
propan-2-yl 4-chloro-3-({[1-(4-methyl-1H-imidazol-2-yl)propyl]carbamoyl}amino)benzoate
phenyl(1-{[1-(pyrimidin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanamide