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3-ethyl-1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperidine-3-carboxylic acid
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-{1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}pyridine
N-cyclopropyl-3-[5-(2-hydroxy-3-methylbenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
N-{5-[1-(furan-2-ylmethyl)-1H-imidazol-2-yl]pyrimidin-2-yl}benzenesulfonamide
3-(2-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)-2,3-dihydro-1λ6-thiophene-1,1-dione
4-{[1-(2-fluorophenyl)propan-2-yl]amino}-N,N-dimethylbutanamide
1-[3-(2-fluorophenyl)-1H-pyrazole-4-carbonyl]-N-phenylpiperidin-3-amine
methyl[(3-{[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl][2-(1H-1,2,4-triazol-1-yl)ethyl]amine
7-fluoro-3-({[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}methyl)-1,2-dihydroquinolin-2-one
2-(2-phenyl-1H-imidazol-1-yl)-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]acetamide
1-[3-(propan-2-yl)adamantan-1-yl]-3-(1,3,4-thiadiazol-2-yl)urea
3-({4-[(2-fluorophenyl)methyl]piperazin-1-yl}methyl)pyrrolidin-3-ol
4-ethyl-3-({1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1'-{[4-(1H-imidazol-1-yl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(4aR,7aS)-1-ethyl-4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N4-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-2-methylpyrimidine-4,6-diamine
2-[1-(5-ethyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
5,7-dimethyl-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-fluoro-N-{1-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
5-(1-benzofuran-2-yl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2-methoxyphenyl)methyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
4-fluoro-2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenol
1-(adamantan-2-yl)-3-(2H-1,3-benzodioxole-5-carbonyl)piperidine
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]propanamide
4-acetyl-N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-{[4-(3-chlorophenyl)-5-(pyrazin-2-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(2R)-1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxy-2-phenylethan-1-one
1-[3-(3,4-dimethoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-4-methylpiperidine
ethyl 1-[1-(3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)piperidin-4-yl]piperidine-3-carboxylate
4-phenyl-1-{spiro[2.2]pentane-1-carbonyl}piperidine-4-carbonitrile
2-[4-({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}amino)-6-methylpyrimidin-2-yl]phenol
1-(3-hydroxypropyl)-4-(1H-1,2,4-triazole-5-carbonyl)-1,4-diazepan-6-ol
N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl 5-[(butan-2-yl)amino]-1-[2-(1H-indol-3-yl)ethyl]-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(5-{[1-(propan-2-yl)piperidin-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)phenol
N-({7-[(2E)-3-(2,5-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
4-{1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methylphenyl)methyl]acetamide
({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[2-(4-methylphenoxy)ethyl]amine
1-(6-aminohexanoyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
6-[2-(4-fluorophenoxy)ethyl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile
N-butyl-4-{[2-(1H-indol-3-yl)ethyl]amino}-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
4-hydroxy-N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-4-hydroxy-N-methyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
methyl 5-{[(2,3-difluorophenyl)methyl]amino}-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea