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N-[(3R,4S)-1-[(3-methylpyridin-2-yl)methyl]-4-propylpyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
3-benzyl-5-(1H-imidazol-4-ylmethyl)-1H-1,2,4-triazole
2,2-diphenyl-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
6-[4-(3-phenylpropyl)piperazin-1-yl]pyrimidine-2,4-diamine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(3-methoxyphenyl)-N-methyl-1,3-benzoxazole-6-carboxamide
(3S,4R)-1-[(5,7-dimethyl-2,1,3-benzoxadiazol-4-yl)sulfonyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
(1S,9aR)-1-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-octahydro-1H-quinolizine
3-(2-methoxyphenyl)-3-[2-(3-methoxypiperidin-1-yl)-2-oxoethyl]-1-methylpyrrolidine-2,5-dione
2-(1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-2-yl)acetamide
3-{[1-(2-methanesulfonylethyl)pyrrolidin-3-yl]methyl}benzoic acid
N-(2-methoxyethyl)-3-[(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)oxy]benzamide
N-(furan-2-ylmethyl)-2-{3-[3-(2-methylpyrimidin-4-yl)phenyl]-1H-pyrazol-1-yl}acetamide
methyl (2S)-1-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidine-2-carboxylate
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-(oxan-4-yl)urea
3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]urea
3-(2-methoxyphenyl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
5-methoxy-N,1-dimethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole-2-carboxamide
N-{[3-(dimethylamino)phenyl]methyl}-4-(4-methylphenoxy)piperidine-4-carboxamide
(1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-3-(2-phenoxyethyl)piperidin-3-yl)methanol
1-(4-methoxyphenyl)-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-3-(propan-2-yl)-1H-1,2,4-triazole
N-[2-(1-{2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxybenzoyl}piperidin-2-yl)ethyl]acetamide
methyl 7-oxo-9-(thiophen-3-ylmethoxy)-3-{[3-(trifluoromethyl)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(2R,3R)-1'-butanoyl-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
5-(azepane-1-carbonyl)-1-benzyl-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
5-{1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-imidazol-2-yl}-2-(pyrrolidin-1-yl)pyrimidine
N-{4-methoxy-3-[2-(pyridin-4-yl)-1H-imidazol-1-yl]phenyl}acetamide
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(3S,4R)-1-(1,3-dihydroxypropan-2-yl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
3-(5-methylfuran-2-yl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
2,4-dimethyl-5-[3-(1H-pyrazol-3-yl)phenyl]-1,3-thiazole
5-methyl-1'-(5-phenyl-1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[3-(1H-pyrazol-1-yl)phenyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
2-[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-5-methylpyrazine
4-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}benzoic acid
5-chloro-N-(1-hydroxypropan-2-yl)-N-methyl-3-phenyl-1H-indole-2-carboxamide
4-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-6-methylpyrimidin-2-amine
methyl 5-[(cyclohex-3-en-1-ylmethyl)amino]-1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-methyl-N-[1-(pyridin-2-yl)propan-2-yl]thian-4-amine
4-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N,6-dimethylpyrimidin-2-amine
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
2-{1-[(4-methylphenyl)methyl]-4-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-yl}ethan-1-ol
5-(1H-1,3-benzodiazol-1-yl)pyridin-2-ol
N-{1-[({[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}-4-oxo-4-phenylbutanamide
2-methyl-4-(4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenyl)butan-2-ol
4-{2,8-diazaspiro[4.5]decan-2-ylmethyl}-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
1-[5-(1-ethyl-1H-indol-6-yl)-4-phenyl-1H-imidazol-1-yl]-3-methoxypropan-2-ol
4-cyclobutyl-6-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrimidin-2-amine
N-(3-butanamidophenyl)-4-(3-oxo-3,4-dihydropyrazin-2-yl)piperazine-1-carboxamide
3-(2-ethylphenoxy)-N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)azetidine-1-carboxamide