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8-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-phenoxy-N-[4-(4-{[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
1-[2-(cyclohex-1-en-1-yl)ethyl]-3-(5-methanesulfonamido-2-methylphenyl)urea
5-(3-methoxyphenoxymethyl)-N-(oxan-4-yl)-1,2-oxazole-3-carboxamide
1-[(2-fluorophenyl)methyl]-N-(isoquinolin-5-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-[2-methoxy-5-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
4-[1-benzyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]-1-methylpiperidin-4-ol
1-[(3-fluorophenyl)methyl]-5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
N-(oxolan-2-ylmethyl)-5-(thiomorpholin-4-ylmethyl)pyrimidin-2-amine
4-(hydroxymethyl)-1-(pyridin-4-ylmethyl)azepan-4-ol
N-(3-hydroxypropyl)-1-{1-[(3-phenoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
methyl 1-({4-[4-(4-methoxyphenyl)-4-oxobutanoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
4-[1-(3,5-dimethoxybenzoyl)piperidin-4-yl]-5-phenyl-2-(pyridin-3-yl)pyrimidine
4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]quinoline
2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
N-[(3,5-dimethoxyphenyl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
3-(2,5-difluorobenzoyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine
1-{3-[4-(naphthalen-1-yl)-1H-pyrazol-5-yl]piperidin-1-yl}pent-4-en-1-one
(3aS,7aR)-5-methyl-2-(5-methylpyrazine-2-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-{[1-cyclohexyl-3-(cyclopropylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]formamido}-N-methylacetamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
4-({5-[1-(cyclopropylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-benzyl-2-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]acetamide
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-N-(pyridin-3-ylmethyl)-2-(trifluoromethyl)benzamide
N-(2-{4-[(3-cyclopentylpropanamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)-3-phenoxypropanamide
5-fluoro-6-methyl-2-(2-{[4-(pyridin-4-ylmethyl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-{3-[(4-methylphenyl)sulfanyl]propyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-[4-(4-methoxyphenyl)piperazin-1-yl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
1-[(4-fluorophenyl)methyl]-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methyl-1H-pyrazole-3-carboxamide
N-[2-(dimethylamino)ethyl]-4-methoxy-3-({1-[(2-methylphenyl)methyl]piperidin-4-yl}oxy)benzamide
1-[2-(4-methoxyphenyl)acetyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
N,N-diethyl-2-{[(furan-3-ylmethyl)(methyl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-(cyclohexylmethyl)-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}benzamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(oxolane-3-carbonyl)piperidine
2,5-dimethoxy-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzene-1-sulfonamide
2-[1-(2,2-dimethylpropyl)-4-(1H-pyrazol-3-ylmethyl)piperazin-2-yl]ethan-1-ol
3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}propanamide
N-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}(2H-1,3-benzodioxol-5-ylmethyl)amine
1-ethyl-N-{2-[methyl(phenyl)amino]propyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(3R,4S)-1-[(2-cyanophenyl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
ethyl 2-(1-{1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidin-3-yl}-N-methylformamido)acetate
9-[(2,3-difluoro-4-methylphenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-benzyl-N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-1,3-thiazole-4-carboxamide
N-[2-(2-fluorophenyl)-1-[1-(2-phenoxypropanoyl)piperidin-4-yl]ethyl]-N-methylthiophene-3-carboxamide
N-(3-phenylpropyl)-6-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
1-[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine