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(4aR,8aS)-1-[2-(2-fluorophenyl)ethyl]-6-(2-methoxybenzoyl)-decahydro-1,6-naphthyridin-2-one
2-(morpholin-3-yl)-N-[4-(1H-1,2,4-triazol-1-yl)phenyl]acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-5-({[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}methyl)-1H-1,2,4-triazole
methyl 1-(benzyloxy)-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
(3S)-N,N-dimethyl-1-(2,4,5-trimethoxybenzoyl)azepan-3-amine
5-(1-cyclopentanecarbonylpiperidin-4-yl)-3-[(4-fluorophenyl)methyl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-(1,2-diethyl-1H-1,3-benzodiazol-5-yl)-2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carboxamide
(2E)-3-(2-fluorophenyl)-N-{[3-methyl-7-(1,3-thiazole-5-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}prop-2-enamide
2-{2-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-1H-imidazole
3-ethynyl-N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)benzamide
N-[5-({4-[4-ethyl-1-(2-methylprop-2-en-1-yl)-2,5-dioxoimidazolidin-4-yl]piperidin-1-yl}methyl)thiophen-2-yl]acetamide
4-{4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanoyl}-1-phenylpiperazin-2-one
4-{5-[(1-propyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}quinoline
N-(1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
1-[(3S,4R)-1-[4-(benzyloxy)butanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-{[7-fluoro-5-(3-fluoro-4-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
3-methyl-1-(2-methylpropyl)-8-{[4-(trifluoromethoxy)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(methyl)(quinolin-5-ylmethyl)amine
ethyl 1-(2-benzyl-1,3-benzoxazole-5-carbonyl)piperidine-3-carboxylate
1-[(8-methoxy-2H-chromen-3-yl)methyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,5-dimethylbenzamide
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[3-(morpholin-4-yl)propyl]propanamide
N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(diphenylmethyl)-1,2-oxazole-5-carboxamide
(4aR,8aS)-1-cyclohexanecarbonyl-N,N-dimethyl-decahydro-1,6-naphthyridine-6-sulfonamide
[3-({1-[2-methyl-2-(morpholin-4-ylmethyl)propyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
[4-(3-phenyl-1,2,4-oxadiazol-5-yl)-1,4-oxazepan-6-yl]methanol
4-[(3,4-dimethoxyphenyl)methyl]-3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
(1R)-1-[1-(1-methylpiperidin-4-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethan-1-amine
(3S,4S)-1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-3,4-diol
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)propanamide
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-2-methyl-N-[(3S)-2-oxoazepan-3-yl]-1,3-thiazole-4-carboxamide
(4aS,7aR)-1-[(3-hydroxyphenyl)methyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]benzonitrile
N-(3,5-dimethylphenyl)-3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
5-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
3,5-dimethyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1,2-oxazole-4-carboxamide
N-benzyl-2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methylacetamide
methyl 3-(2-chlorobenzoyl)-9-[2-(2-fluorophenyl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3-(2-oxoimidazolidin-1-yl)benzamide
(2R,3R,6R)-3-phenyl-5-(quinoxalin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2-oxo-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,2-dihydropyridin-2-one
methyl 5-[(2,2-dimethylpropyl)amino]-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-({1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-5-(methoxymethyl)-N-[(3S)-2-oxoazepan-3-yl]furan-2-carboxamide
3-[(4aR,7aS)-4-(1H-indol-5-ylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
(2S,4S)-4-[2-(2,3-dihydro-1H-inden-5-yloxy)-2-methylpropanamido]-N-ethyl-1-methylpyrrolidine-2-carboxamide