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2-hydroxy-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-4-(methylsulfanyl)butan-1-one
1-{3-[({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]piperidin-1-yl}ethan-1-one
6-{[5-oxo-1-(propan-2-yl)pyrrolidin-3-yl]amino}pyridine-3-carbonitrile
4-{6-[4-(1-ethoxyethyl)phenyl]pyridazin-3-yl}thiomorpholine
6-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-N,N-dimethylpyridine-2-carboxamide
4-[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]-1-[(2R)-oxolane-2-carbonyl]piperidine
6-(cyclopropylmethoxy)-4-(2-methyl-1,3-thiazole-4-carbonyl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N-[(3R,4R)-3-hydroxy-1-[6-methyl-2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-yl]pyridine-2-carboxamide
1-{4-[(3-hydroxyphenyl)methyl]piperazin-1-yl}-2-(1-methylpiperidin-2-yl)ethan-1-one
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[(3-methyloxetan-3-yl)methyl]amine
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-[2-phenyl-1-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)ethyl]pyridine-2-carboxamide
1-(5-methylhex-5-en-2-yl)-4-[2-(piperidin-1-yl)ethyl]-1,4-diazepan-5-one
8-[2-(2,5-difluorophenyl)acetyl]-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
1-methyl-2-(morpholin-4-yl)-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
5-[({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]-N,N-dimethyl-1,3-thiazol-2-amine
ethyl 2-[2-({1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidin-4-yl}formamido)ethyl]-1,3-thiazole-4-carboxylate
N-[(3S)-1-benzylpyrrolidin-3-yl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
4-(4-chloro-1-methyl-1H-indazol-3-yl)-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
3-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
1-(3-{1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}phenyl)imidazolidin-2-one
2-{4-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[(5-chlorothiophen-2-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-({1-[3-(2-methyl-1H-imidazol-1-yl)propyl]piperidin-2-yl}methyl)morpholine
4-(pyridin-3-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-2-amine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
4,5-dimethyl-6-{4-[1-(propan-2-yl)piperidine-3-carbonyl]piperazin-1-yl}pyrimidine
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[3-(methylsulfanyl)propyl]acetamide
1-{2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(furan-2-carbonyl)piperazine
8-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2-(propan-2-yl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
(3S,4R)-1-[(3-carboxyphenyl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-{3-oxo-3-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]propyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(4aS,8aR)-1-benzyl-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
4-fluoro-3-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
2-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]benzoic acid
methyl (2S,4S)-4-(3-chlorobenzamido)-1-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
1-(5-{[3-(hydroxymethyl)-4-methylpiperazin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
10-(3-hydroxypiperidine-1-carbonyl)-9-methoxy-3-[(3-methylthiophen-2-yl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(1H-1,2,4-triazol-1-yl)acetamide
N,N-dimethyl-2-{N-methyl-1-[3-({1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)phenyl]formamido}acetamide
(2S)-2-phenyl-2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)acetamide
2-{[4-(benzyloxy)phenyl]methyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-benzyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1,3-benzoxazole-5-carboxamide
methyl 4-(5-chloro-2-{[3-(3-methyl-1H-pyrazol-1-yl)propanamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
3-[1-(pyridin-4-yl)-1H-imidazol-2-yl]benzoic acid
1-{[1-(2-fluorophenyl)cyclopentyl]methyl}-3-(5-methyl-4H-1,2,4-triazol-3-yl)urea
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]propan-1-one
4-(2-methoxyphenoxy)-1-(pyridin-2-ylmethyl)piperidine-4-carboxylic acid
4-methyl-3-(3-oxo-4-phenylpiperazine-1-carbonyl)benzene-1-sulfonamide