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N-{1-[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-2-carboxamide
5-cyclobutyl-N-[2-(ethanesulfonyl)ethyl]-1,3,4-oxadiazol-2-amine
4-(1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)thiomorpholine
1-phenyl-4-{[2-(thiophen-2-yl)azetidin-1-yl]methyl}-1H-1,2,3-triazole
(1H-imidazol-2-ylmethyl)(methyl)[(3-methyl-1H-indol-2-yl)methyl]amine
4-chloro-1,5-dimethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1H-pyrazole-3-carboxamide
N-ethyl-5-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
8-[(2-chlorophenyl)methyl]-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-2-(methylamino)pyridine-3-carboxamide
4-cyclobutanecarbonyl-9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[2-(5-methylfuran-2-yl)phenyl]methyl}amine
4-(2-methoxyphenoxy)-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
1-[3-(2-methylphenoxy)azetidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
4-(4-methylphenyl)-N-[(5-methylpyrazin-2-yl)methyl]-5-(pyridin-4-yl)pyrimidin-2-amine
N-(4-chloro-3-methylphenyl)-2-{[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]amino}acetamide
1-(pent-4-enoyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-[(4-{4-[(2-hydroxyethyl)amino]quinazolin-6-yl}phenyl)methyl]acetamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
(3R,4R)-4-amino-1-(4-methyl-2-phenylpyrimidine-5-carbonyl)piperidin-3-ol
3-[5-oxo-2-(thiophen-3-ylmethyl)pyrrolidin-2-yl]-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]propanamide
5-[(3-methoxyphenyl)methyl]-5-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-3-methylimidazolidine-2,4-dione
2-(3-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenoxy)propanoic acid
5-{[(3S,5R)-1-[(3,4-dimethoxyphenyl)methyl]-5-(pyrrolidine-1-carbonyl)piperidin-3-yl]methoxy}-2-methylpyridine
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-3-methoxypropanamide
4-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-N-(3-hydroxyphenyl)-4-oxobutanamide
{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}acetamide
5-(2,4-difluorophenoxymethyl)-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
3-methyl-7-{[4-(methylsulfanyl)phenyl]methyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-[(2-methoxyethyl)sulfamoyl]-N-methyl-N-(1H-pyrazol-3-ylmethyl)benzamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylspiro[2.3]hexane-1-carboxamide
(2S)-2-[(1-cyclopentanecarbonylpiperidin-4-yl)formamido]-3-phenylpropanoic acid
1-(1-{[3-(2-aminoethyl)phenyl]methyl}piperidin-4-yl)-3-phenylpropan-1-ol
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]acetamide
N-(2,2-dimethylpropyl)-N-ethyl-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
4-[2-(4-fluorophenyl)azetidine-1-carbonyl]-1,2-dihydroquinolin-2-one
3-(1-methylpiperidin-3-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-1-methyl-1H-pyrazole-5-carboxamide
3-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carbonyl)pyridine
5-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-2,1,3-benzoxadiazole
1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxypropyl)piperidine
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(4S)-1-(4-chloro-1-ethyl-1H-pyrazole-5-carbonyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
2-methoxy-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)acetamide
5-{[(5-chlorothiophen-2-yl)methyl]amino}-1-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(3-methoxyphenyl)-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-{4-[5-phenyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1H-indole
4-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H-imidazole-5-carboxamide
3-methyl-1-(2-methylpropyl)-8-(oxan-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-ethyl-1-methyl-4-[3-(pyridin-3-yl)propanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one