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(2E)-N-({3-methyl-7-[(2E)-4-methylpent-2-enoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenylprop-2-enamide
3-(4-phenyl-1H-pyrazol-5-yl)piperidine
(2R)-2-amino-3-hydroxy-1-[2-({methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]propan-1-one
1-[(2-aminopyridin-3-yl)methyl]-3-[(dimethylamino)methyl]piperidin-3-ol
5-[2-(3,4-dimethoxyphenyl)ethyl]-3-(2-methylpropyl)-1H-1,2,4-triazole
4-{6-[1-(4-methylpyridine-3-carbonyl)piperidin-3-yl]pyrimidin-4-yl}morpholine
N-[3-(3-chlorophenyl)phenyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidine-4-carboxamide
3-(3-fluorophenyl)-4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperazin-2-one
N-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]thiophene-2-carboxamide
(2S,4R)-4-[4-(4-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}phenyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]acetamide
3-[(2-chlorophenyl)methyl]-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(diphenylmethyl)-2-ethyl-6-methyl-4-oxo-1-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
9-[4-(1H-imidazol-1-yl)butanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopentyl-5-(4-methylbenzoyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-(2,4-difluorophenyl)-1-(1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}piperidin-4-yl)ethyl]-N-methylcyclopropanecarboxamide
N-{[7-(5-chloro-3-methyl-1H-indole-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}oxolane-2-carboxamide
1-(1,3-dioxo-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindol-4-yl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxamide
2-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]morpholin-3-yl}acetic acid
2-(2,5-dioxoimidazolidin-1-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}acetamide
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}propanamide
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-3-phenyl-1,2-oxazole-5-carboxamide
(1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
4-(1-hydroxy-3-methylbutan-2-yl)-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
3-methoxy-N-(1-{7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
(3R,4R)-1-(1,3-benzothiazol-2-yl)-3-cyclopropyl-4-methylpyrrolidin-3-ol
9-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-3,9-diazaspiro[5.5]undecane-2,4-dione
4-{[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
3-(3-methoxyphenyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-3-(1,3,4-thiadiazol-2-yl)urea
2-[2,4-dimethyl-6-(pyridin-4-yl)phenoxy]acetic acid
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(1H-indazol-1-yl)acetamide
6-(benzyloxy)-4-[3-(methylsulfanyl)propanoyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
4-[2-oxo-2-(piperidin-1-yl)ethoxy]-N-[2-(2-oxopyrrolidin-1-yl)ethyl]benzamide
1-{[4-(cyclopentyloxy)phenyl]methyl}-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
2-{2-methylimidazo[1,2-a]pyridin-3-yl}-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)acetamide
N-(1-benzothiophen-5-ylmethyl)-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
3-{5-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
3-(5-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
3-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
3-(3,4-dimethoxybenzoyl)-1-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]piperidine
1-{2-hydroxy-3-[4-methoxy-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxy]propyl}piperidin-4-ol
N-[2-(4-fluorophenyl)-1-{1-[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetyl]piperidin-4-yl}ethyl]-2-methoxy-N-methylacetamide
2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)-N-propylacetamide
N-({2-[(dimethylamino)methyl]phenyl}methyl)-N-methylpyrimidin-2-amine
6-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-2,3,4,5-tetrahydropyridazin-3-one
3-(3-methoxyphenyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
N-[3-(2-methylquinolin-5-yl)phenyl]acetamide
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide