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methyl 1-(benzyloxy)-8-(cyclopropylmethyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
3-(2-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-2-oxoethyl)-1,3-thiazolidine-2,4-dione
1-(3-hydroxy-1,2-oxazole-5-carbonyl)-4-[(2-methoxyphenyl)methyl]-1,4-diazepan-6-ol
N-(3-ethoxy-2-hydroxypropyl)-5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
N-methyl-2-(pyridin-2-yl)-N-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[1'-(dimethyl-1,2-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
5-[1-(1H-imidazol-2-ylmethyl)-1H-1,2,3-triazol-4-yl]quinoline
N-[1-(furan-2-carbonyl)piperidin-3-yl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
(2S)-2-{2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]acetamido}-4-methylpentanamide
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-dichlorobenzamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-(dimethylamino)ethyl]-3-{2-[(2S)-4-methyl-2-phenylpiperazin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
(3S,4S)-1-(4-fluorobenzoyl)-4-(naphthalen-2-yl)piperidin-3-ol
N-[1-(furan-2-yl)ethyl]-3-(2-methoxyphenyl)-N-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-(propan-2-yl)furan-3-carboxamide
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]propan-1-one
1-(cyclopropylmethyl)-4-(3-methanesulfonylbenzoyl)-2-(propan-2-yl)-1,4-diazepane
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-[2-(pyridin-3-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(5-ethylpyridin-2-yl)methyl]-1-[(3-methoxyphenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
1-[2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(methoxymethyl)piperidine
3-(naphthalene-2-carbonyl)-1-phenylmethanesulfonylpiperidine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-cyclopropyl-N-(pyridin-3-ylmethyl)acetamide
1-(2,3-dichlorophenyl)-3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]urea
2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-4-(5-methanesulfonyl-2-methylpyrimidin-4-yl)morpholine
1-benzyl-3-(2-methylpropyl)-8-(oxan-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(butan-2-yl)-N3-ethyl-4-oxo-N5-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
5-[3-(2-methylpropanamido)pyridin-2-yl]thiophene-2-carboxylic acid
N-cyclopropyl-3-[5-(2-phenylethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-(4-methoxyphenyl)-4-[1-(oxan-4-yl)piperidin-3-yl]piperazine
(3R,4S)-1-(1-cyclobutanecarbonylpiperidin-4-yl)-4-cyclopropylpyrrolidin-3-amine
5-(4-benzylpiperidin-1-yl)-1-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(butan-2-yl)({[4-methoxy-3-(methoxymethyl)phenyl]methyl})(pyridin-4-ylmethyl)amine
2-(adamantan-1-yl)-4-hydroxy-N-[2-(pyrazin-2-yl)ethyl]pyrimidine-5-carboxamide
N-[(3-methoxyphenyl)methyl]-3-[1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]propanamide
N-[(1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]acetamide
N-[2-(4-chlorophenyl)-2-hydroxyethyl]-2-(1-ethylpiperidin-4-yl)acetamide
N-[(5-fluoro-2,3-dimethyl-1H-indol-7-yl)methyl]-3-(1,2-oxazolidin-2-yl)propanamide
7-oxo-N-[1-(3-phenylpropyl)piperidin-3-yl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
1-(cyclohexylmethyl)-5-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazole
5-acetamido-2-ethyl-N-methyl-1-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
3-[(2,3-dimethoxyphenyl)methyl]-5-methyl-5-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-4-amine
3-({[(2-chlorophenyl)methyl]amino}methyl)-1-(cyclohexylmethyl)-6,7-dimethoxy-1,2-dihydroquinolin-2-one
N-[(3R,4S)-4-cyclopropyl-1-(3-methoxypropanoyl)pyrrolidin-3-yl]methanesulfonamide
9-(2-methoxypyridine-3-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
{3-[(2-fluorophenyl)methyl]-1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperidin-3-yl}methanol
4-({1-[(4-methoxypyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
ethyl 4-(cyclopropylmethyl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperidine-4-carboxylate