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1,3-dimethyl-6-{3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
1-(cyclohexylmethyl)-5-[4-(2-hydroxyethyl)piperazin-1-yl]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}methanesulfonamide
N-methyl-4-(quinolin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-{[(benzylsulfamoyl)(methyl)amino]methyl}phenol
N-[(3,5-dimethoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-2-(methylsulfanyl)acetamide
1-(1,3-benzothiazol-2-yl)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]piperidin-4-amine
1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
3-methyl-N-[(1R,3S)-3-[(2,2,2-trifluoroethyl)carbamoyl]cyclopentyl]-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
2-(1-tert-butyl-1H-pyrrole-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-[2-(piperidin-2-yl)ethyl]-5-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]phenol
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-5-propyl-1,3,4-oxadiazole-2-carboxamide
methyl 4-{[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}butanoate
3-(1H-indol-3-yl)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
3-methyl-4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
5-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-3-oxopropyl}-5-[(4-chlorophenyl)methyl]pyrrolidin-2-one
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[4-(1-hydroxypropyl)piperidin-1-yl]ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[1-(pyridin-2-yl)propan-2-yl]amino}piperidin-1-yl)benzamide
3-chloro-2-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]-5-(trifluoromethyl)pyridine
N-methyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
7-(4-chloro-1H-pyrazole-3-carbonyl)-N,N-dimethyl-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(dimethylamino)-N-{3-methyl-1-[7-(4-oxo-4-phenylbutanoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}acetamide
7-(1-phenylcyclopropanecarbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
(1R,5S,6R)-3-[(2-hydroxy-5-methoxyphenyl)methyl]-N-[(5-methylpyrazin-2-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3-(piperidin-3-yl)benzamide
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-{2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}acetamide
N-ethyl-6-[(1,4-oxazepan-6-ylmethyl)amino]pyridine-3-carboxamide
4-(3,5-dimethylfuran-2-carbonyl)-2-[(4-fluorophenyl)methyl]morpholine
9-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[3-(1H-imidazol-1-yl)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-3-yl)pyrrolidin-2-one
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
(3S,4R)-4-(3-methoxyphenyl)-1-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
(furan-3-ylmethyl)(methyl)({5-[(oxolan-2-ylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)amine
N-{[7-(5-chloro-2-fluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
3-[1-(6-cyanopyridin-2-yl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
(3R,4R)-4-(hydroxymethyl)-1-{[3-(pyridin-2-yl)phenyl]methyl}piperidin-3-ol
3-(4-fluorophenyl)-N-[3-(4H-1,2,4-triazol-4-yl)propyl]-1H-pyrazole-5-carboxamide
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
1-(3,5-dichloro-4-methylbenzoyl)-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
5-(2-chlorophenyl)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-2-methylfuran-3-carboxamide
4-[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-2-(2-methoxyethyl)morpholine
1-{3-[2-({[(4-ethylphenyl)methyl](methyl)amino}methyl)-4-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
5-{1-[2-(2,6-difluorophenyl)acetyl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
4-(4-cyclobutyl-6-methylpyrimidin-2-yl)-1,4-oxazepan-6-ol
[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl](pyridin-3-yl)methanol
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]methanol