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ethyl 1-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-5-{[(1-methoxypropan-2-yl)amino]methyl}-1H-pyrazole-4-carboxylate
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1-(4,6-dimethylquinazolin-2-yl)piperidine-4-carboxamide
N-({7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2,6-difluorobenzamide
3-{3-oxo-3-[2-(pyridin-2-yl)piperidin-1-yl]propyl}-3,4-dihydroquinazolin-4-one
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-1-(morpholin-4-yl)ethan-1-one
3-(3-methylphenoxy)-1-{spiro[2.3]hexane-1-carbonyl}azetidine
6-(4-chlorophenyl)-N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-cyclohexyl-N3-[(2-methoxynaphthalen-1-yl)methyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-[4-(ethanesulfonyl)piperazin-1-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene
5-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-pyrazol-3-yl]-N-[(4-methoxyphenyl)methyl]-4-methyl-1,3-thiazol-2-amine
4-{4-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(2-methoxyethyl)-2,3-dihydro-1H-isoindole-1,3-dione
8-(1-aminocyclopropanecarbonyl)-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-(2,3-dihydro-1H-inden-2-yl)-8-{[4-(furan-2-yl)phenyl]methyl}-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-phenoxy-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
ethyl 4-({3-[benzyl(methyl)amino]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
4-[4-(2-chlorophenoxy)piperidine-1-carbonyl]-1-ethylpyrrolidin-2-one
methyl 4-[4-(oxolan-3-ylmethyl)piperazin-1-yl]benzoate
1-(4-ethylpiperazin-1-yl)-3-[3-({[(5-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
ethyl 4-[1-(5-phenylpentanoyl)piperidin-3-yl]piperazine-1-carboxylate
4-(1H-1,3-benzodiazol-2-yl)-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
5-[(2-fluoro-4-methoxyphenyl)methyl]-5-{3-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
6-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine-2,4-diamine
4,4,4-trifluoro-1-{3-[5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
2-[(3S,4R)-3-acetamido-4-propylpyrrolidin-1-yl]-N-[2-(4-fluorophenyl)ethyl]acetamide
1-(3-chlorophenyl)-4-(5-methoxyfuran-2-carbonyl)-5-methylpiperazin-2-one
N-[(1-benzylpyrrolidin-3-yl)methyl]-5-hydroxy-4-oxo-4H-pyran-2-carboxamide
N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)propanamide
N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanamide
5-(2-fluorophenyl)-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-1,2,4-triazin-3-amine
2-[6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
2-{[2-(trifluoromethyl)morpholin-4-yl]methyl}-1,4-dihydroquinolin-4-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-(cyclopropylmethyl)-1-(propan-2-yl)-1H-pyrazole-3-carboxamide
3-[2-({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)propyl]-3,4-dihydroquinazolin-4-one
N-({6-[4-(3-chlorophenyl)piperazin-1-yl]-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)-2,2-dimethyloxan-4-amine
4-(2,5-dimethoxyphenyl)-3-methyl-4H-1,2,4-triazole
1-(2-methoxyphenyl)-2,2-dimethyl-4-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperazine
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-(2-methoxyethyl)-8-[(4-methoxyphenyl)methyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,5R)-N-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-2,3,4-trimethoxy-N-(oxolan-2-ylmethyl)benzamide
6-butyl-2-(4-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
4-{[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]carbamoyl}pyridin-1-ium-1-olate
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
2-methyl-1-{4-[4-(propan-2-yl)-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}propan-2-amine
4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-2-amine
2-(4-fluorophenoxymethyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1,3-oxazole-4-carboxamide
(1R,7S)-3-[(3-methoxyphenyl)methyl]-6-(piperidine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one