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[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]({[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl})methylamine
{[(3S,4R)-1-(2-methoxypyridine-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
N-propyl-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-N-(thiophen-3-ylmethyl)acetamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-(piperidin-4-ylmethyl)benzamide
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(6-hydroxy-6-methylheptan-2-yl)benzamide
5-methanesulfonyl-1'-(4-methoxypyrimidin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-methyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-1,2,3-thiadiazole-5-carboxamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-1-(methoxymethyl)cyclobutane-1-carboxamide
6-[2-(phenylsulfanyl)acetyl]-N-(thiophen-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
2-[4-(2-methylpropyl)phenyl]-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(1H-pyrazol-1-yl)benzamide
3-[(4-fluorophenyl)methyl]-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-1,2-oxazole-5-carboxamide
methyl 3-(3-chlorobenzoyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2E)-1-{4-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}-3-(pyridin-4-yl)prop-2-en-1-one
N-(2-{7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
(2S,4R)-N-ethyl-1-(furan-3-ylmethyl)-4-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanamido]pyrrolidine-2-carboxamide
2-(oxane-4-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
9-(5,6-dimethylpyrimidin-4-yl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3,4-difluorophenyl)methyl]-3-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl}propanamide
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2-(4-propanoylphenoxy)acetamide
[2-(3,4-dimethoxyphenyl)ethyl]({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
(4-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}morpholin-3-yl)methanol
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-8-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
4-[2-(3-hydroxyphenyl)-1H-imidazol-1-yl]-2-(pyrrolidin-1-yl)benzamide
9-methoxy-7-oxo-3-[2-(pyridin-3-yl)acetyl]-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[(4-chlorophenyl)methyl]-8-[(2R)-oxolane-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
5-cyclopropyl-N-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-(oxolan-3-yl)-1H-pyrazole-4-carboxamide
4-(4-chlorophenoxy)-1-{3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidine
2-[4-(dimethylamino)azepan-1-yl]pyridine-3-carboxamide
8-chloro-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]quinoline-2-carboxamide
N,N-diethyl-2-({1-[(4-methoxyphenyl)methyl]-2-oxo-4-(propan-2-yl)-1,4-diazepan-6-yl}oxy)acetamide
{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4-(2-phenylethyl)piperidin-4-yl}methanol
1-[2-(4-chlorophenyl)ethyl]-N-{[4-(methylsulfanyl)phenyl]methyl}-6-oxopiperidine-3-carboxamide
1-(1-{2-[4-(methylsulfanyl)phenyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carbonyl)piperidine-3-carboxamide
N-(1-{7-[(2-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
2-methyl-6-(piperidin-4-yl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-4-amine
5-cyclopropanecarbonyl-1'-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-ethyl-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-{imidazo[1,2-a]pyridine-2-carbonyl}-2,7-diazaspiro[4.5]decane
(2S)-2-{[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]formamido}pentanoic acid
1-benzyl-6-(pyridin-3-ylmethoxy)-4-(quinoline-6-carbonyl)-1,4-diazepan-2-one
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-[(2-fluorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-2-propyl-N-(pyridin-4-ylmethyl)-1,3-thiazole-4-carboxamide
4-benzyl-9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N5,N6,N6-trimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-[(4-fluorophenyl)methyl]-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
4-ethyl-3-{1-[6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[1-ethyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(naphthalen-1-ylmethyl)acetamide
(3S,4S)-4-(dimethylamino)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]pyrrolidin-3-ol
2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-5-fluoro-4-(pyrrolidin-1-yl)pyrimidine