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1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-phenylpiperidine-4-carbonitrile
1-(oxane-4-carbonyl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
(3aS,6aS)-2-(2-hydroxyethyl)-5-{[4-(methylsulfanyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{3-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]piperidin-1-yl}-2-[2-(2-methoxyphenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-(3-cyano-4-methoxyphenyl)-3-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
5-fluoro-2-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]-1H-1,3-benzodiazole
1-{2-[(4-methylpiperidin-1-yl)methyl]phenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
4-[4-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)phenyl]-2-methylbutan-2-ol
3-methoxy-4-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)phenol
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-(7-methoxy-4-methyl-2-oxo-2H-chromen-3-yl)acetamide
3-(1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}pyrrolidin-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
{1-[4-(4-{[2-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)benzoyl]piperidin-3-yl}methanol
N-cyclopropyl-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)acetamide
1-(2-methylphenyl)-4-[1-(naphthalene-2-carbonyl)piperidin-3-yl]piperazine
4-(5-chloro-2-methylphenyl)-3-(4-methyl-1H-imidazol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,7aR)-1-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethan-1-one
2-chloro-N-[2-(cyclohex-1-ene-1-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
2-{4-[(dimethyl-1,2-oxazol-4-yl)methyl]-1,4-diazepan-1-yl}-1,3-benzothiazole
(4aS,7aR)-1-(2-chloro-4-fluorobenzoyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-ethyl-2-(2-fluorophenyl)-5-[2-(hydroxymethyl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-7-yl]acetamide
6-[(4-ethoxyphenyl)methyl]-N-(2-methoxyphenyl)-6-azaspiro[2.5]octane-1-carboxamide
2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-{2-[4-(propan-2-yloxy)phenyl]ethyl}acetamide
3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]-N-{spiro[2.5]octan-1-ylmethyl}propanamide
N,N-diethyl-1-{1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
4-{6-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}thiomorpholine
6-ethoxy-2-{3-[4-(2-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-4-methylquinazoline
3-[4-(3,4-diethoxyphenyl)-1H-imidazol-2-yl]piperidine
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
1-(pyridin-2-yl)-N-{[4-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(2,6-dimethylpyridin-4-yl)piperazine
3,4,5-trimethoxy-N-({4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
1-(3-methanesulfonamidophenyl)-3-[2-(propylsulfanyl)ethyl]urea
2-[(2,3-dihydro-1H-inden-2-yl)amino]-N-ethylpropanamide
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-3-yl)ethan-1-one
5-[1-(2,4-difluorobenzoyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
2-{[(2-fluorophenyl)methyl](methyl)amino}-1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
4-(3,5-dimethoxybenzoyl)-6-methyl-1-[2-(methylsulfanyl)phenyl]piperazin-2-one
2-[3-(dimethylamino)propyl]-9-[2-(4-methyl-1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
5-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]piperidin-2-one
N3-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
3-[2-oxo-2-(3-{[(4-phenylphenyl)formamido]methyl}piperidin-1-yl)ethyl]-1,2,3-oxadiazol-3-ium-5-olate
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-ethyl-3-(propan-2-yl)-N-{2-[4-(propan-2-yloxy)phenyl]ethyl}-1H-pyrazole-5-carboxamide
7-methoxy-N-methyl-N-(1,2-oxazol-3-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl[(5-methyl-1H-pyrazol-3-yl)methyl]{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
4-(2H-1,3-benzodioxol-5-ylmethyl)-7-(3,4-dihydronaphthalen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(methoxymethyl)-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]furan-2-carboxamide
N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide