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3-[2-(4-cyclopentyl-3-oxopiperazin-1-yl)-2-oxoethyl]-3-(3-fluorophenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
7-{[3-(2-methylphenyl)phenyl]methyl}-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-benzyl-6-(cyclopropylmethoxy)-4-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-1,4-diazepan-2-one
1-[(1S,5R)-6-(3-chloro-2-methylbenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-[4-(1-benzothiophen-2-ylmethyl)morpholin-2-yl]ethan-1-amine
N-[4-(4-{[(3-chlorophenyl)methyl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
1-(5-chloro-2-methoxyphenyl)-3-cyclopropyl-5-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-1,2,4-triazole
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2,6-dimethylquinoline-4-carboxamide
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl][(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]amine
methyl 3-(4-{[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(oxan-4-ylmethyl)acetamide
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
3-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
3-(1,2-oxazolidin-2-yl)-N-(pyridin-4-ylmethyl)propanamide
N-{[1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]methyl}-3-(trifluoromethyl)benzamide
methyl 3-(2-methoxybenzoyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-{4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-1,2-benzothiazole
3-[4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-2,5-dimethylpyrazine
N-(4,6-dimethylpyridin-2-yl)-5-[1-(oxan-4-yl)pyrrolidin-2-yl]thiophene-2-carboxamide
methyl 4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperazine-1-carboxylate
2-(ethylamino)-N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)pyrimidine-5-carboxamide
8-(1,3-benzoxazol-2-yl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
8-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[1-(2-chlorobenzoyl)piperidin-3-yl]-4-(4-methoxyphenyl)piperazine
1-[(3-chlorophenyl)methyl]-3-(propan-2-yl)-5-(4H-1,2,4-triazol-4-ylmethyl)-1H-1,2,4-triazole
1-{2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}-N,N-diethylpiperidine-3-carboxamide
methyl (2S,4S)-4-cyclohexaneamido-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxylate
3-benzyl-5-[(2-fluorophenyl)methyl]-1H-1,2,4-triazole
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-ethylphenyl)methyl]-N-methylacetamide
1-{6-[3-(methoxymethyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}azepane
3-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-(3-fluorophenyl)urea
6-methyl-2-propyl-N-[2-(pyridin-2-yl)ethyl]pyrimidin-4-amine
1-(4-ethylphenyl)-3-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}urea
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(5-methoxy-1H-indol-2-yl)methyl]acetamide
(2R,3R,6R)-5-benzoyl-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(3R,4S)-1-(carbamoylmethyl)-4-cyclopropylpyrrolidin-3-yl]-2-(3-methoxyphenoxy)acetamide
[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
8-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}quinoline
(2E)-3-(4-methoxyphenyl)-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)prop-2-enamide
benzyl[(2-chloropyridin-3-yl)methyl]methylamine
(4aS,8aR)-6-(1H-1,3-benzodiazol-2-ylmethyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
6-(2-fluorophenyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{[1-(5-hydroxypyrazine-2-carbonyl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
2-[4-(1-benzothiophen-3-yl)-2-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy]-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
(3S,4R)-4-(4-fluorophenyl)-1-(1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
3-(1-butyl-1H-imidazol-2-yl)-N-(2-methylphenyl)piperidine-1-carboxamide
N-[2-(3-methoxyphenyl)ethyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
N-cyclopropyl-1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)piperazine-2-carboxamide
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
(1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-2-phenylethyl)(methyl)(pyridin-3-ylmethyl)amine