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methyl (2S)-1-[1-(4,7-dimethylquinazolin-2-yl)piperidine-3-carbonyl]pyrrolidine-2-carboxylate
N-[(2R,3R)-2-methoxy-1'-(5-methyl-1H-indole-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
5-({[3-fluoro-5-(trifluoromethyl)phenyl]methyl}amino)-1-methyl-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-{5-[(2,4-dioxoimidazolidin-1-yl)methyl]-3-methyl-1H-1,2,4-triazol-1-yl}-4-fluorobenzene-1-sulfonamide
N-[3-(methylsulfanyl)propyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3R,4R)-1-({4-amino-6-[(3-methylphenyl)amino]-1,3,5-triazin-2-yl}methyl)-4-ethylpiperidine-3,4-diol
{[5,8-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}[1-(thiophen-2-yl)ethyl]amine
6-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrazine-2-carboxamide
1-[(3R,4R)-4-(azepan-1-yl)-3-hydroxypiperidin-1-yl]-3-(1H-indol-3-yl)propan-1-one
5-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,1,3-benzoxadiazol-1-ium-1-olate
1-(4-fluorophenyl)-4-{1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}piperazine
2-{5-[(3-methyl-1H-pyrazol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-1,3-benzodiazole
N-[(3S,4R)-1-[(5-chloro-2,4-dimethoxyphenyl)methyl]-4-propylpyrrolidin-3-yl]acetamide
N-cyclopentyl-1-(2-methylpropyl)-5-[3-(1H-pyrazol-1-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-2-yl}pyridine
N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(5-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}furan-2-yl)methanol
4-{3-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
2-[1-(2,2-dimethylpropyl)-4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl]ethan-1-ol
N-(1-{7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)oxolane-3-carboxamide
1-[1-(2-methylbutyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-4-carboxamide
1-[1'-(2-acetylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
2-ethoxy-6-{[methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amino]methyl}phenol
3-hydroxy-N-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
1-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
5-[3-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-oxopropyl]-5-[(2-fluoro-5-methoxyphenyl)methyl]pyrrolidin-2-one
2-(3-{[3-(2-methoxybenzoyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2-(ethylsulfanyl)-5-({2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)pyrimidine
N-[(2S)-2-hydroxypropyl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
2-methyl-3-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
8-(3-ethyl-1H-indole-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-methyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(3-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}propyl)morpholine
(3R)-1-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-3-methylpiperazine
2-(dimethylamino)-2-(2-methylphenyl)-1-[4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
5-ethyl-3-[2-(4-methoxyphenyl)ethyl]-5-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
1-{3-oxo-3-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(2-{2-azabicyclo[2.2.1]heptan-2-yl}-2-oxoethyl)-1-ethyl-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
4-(6-ethylpyrimidin-4-yl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
methyl (2S,4S)-4-(5-amino-4-phenyl-1H-pyrazole-3-amido)-1-methylpyrrolidine-2-carboxylate
N-[3-(furan-2-yl)propyl]-2,6-dihydroxybenzamide
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-3-ol
N-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
methyl 6-[2-(cyclohex-1-en-1-yl)acetyl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
8-(2,3-dihydroxypropyl)-3-{2-[methyl(2-methylpropyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1-benzylpiperidin-4-yl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide