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N-[(E)-N'-(4,6-dimethylpyrimidin-2-yl)-N-[2-(1H-indol-3-yl)ethyl]carbamimidoyl]-3,4,5-trimethoxybenzamide
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-2-[(3S)-3-methyl-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-1-yl]acetamide
(4R)-N-[1-(2-methoxyethyl)-1H-indol-4-yl]-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R,16S)-5,9,16-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentanamide
(4R)-N-(1,3,4-thiadiazol-2-yl)-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R,16S)-5,9,16-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentanamide
2-[(2,2-dimethyl-4-oxo-3,4-dihydro-2H-1-benzopyran-7-yl)oxy]-N-[6-(1H-indol-4-yloxy)pyridin-3-yl]acetamide
2-(2-methylpropyl)-4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1,2-dihydroisoquinolin-1-one
3-(2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl)-N-(5-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}pentyl)propanamide
methyl 2-[(4R)-4-[(1S,2S,5R,7R,10R,11S,14R,15R,16S)-5,16-dihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentanamido]-5-(2-methylpropyl)-1,3-thiazole-4-carboxylate
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
2-(2-methylpropyl)-4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,2-dihydroisoquinolin-1-one
(1Z,4E)-1-hydroxy-5-(1H-indol-3-yl)-1-phenylpenta-1,4-dien-3-one
2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]-N-(3-acetamidophenyl)acetamide
2-[(1,6-dimethyl-4-oxo-1,4-dihydropyridin-3-yl)oxy]-N-[2-(1H-indol-3-yl)ethyl]acetamide
4-(heptan-3-yl)-3-methyl-1-(9H-purin-6-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
ethyl 3-(4-hydroxy-3-methoxyphenyl)-3-(4-hydroxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)propanoate
N-(3-acetylphenyl)-2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]acetamide
methyl (2S)-4-methyl-2-[3-(3-oxo-3,4-dihydroquinoxalin-2-yl)propanamido]pentanoate
ethyl 3-(4-hydroxy-2-oxo-1,2-dihydroquinolin-3-yl)-3-(4-hydroxy-3,5-dimethoxyphenyl)propanoate
3-methyl-4-(propan-2-yl)-1-(9H-purin-6-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[(3R)-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl]-N-[2-(5-fluoro-1H-indol-3-yl)ethyl]acetamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
(4R)-1-(4-benzylpiperazin-1-yl)-4-[(1S,2S,5R,7R,10R,11S,14R,15R,16S)-5,16-dihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentan-1-one
N-(7-methoxyquinolin-3-yl)-2-(1-methyl-1H-indol-3-yl)acetamide
N-[2-(5-methoxy-1H-indol-1-yl)ethyl]-2-(7-methoxy-4-methyl-2-oxo-2H-chromen-3-yl)acetamide
2-[(2S)-1-[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]-1-oxopropan-2-yl]-2,3-dihydro-1H-isoindol-1-one
ethyl 3-(4-hydroxy-3,5-dimethoxyphenyl)-3-(4-hydroxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)propanoate
(4R)-N-[4-(pyridin-2-yl)-1,3-thiazol-2-yl]-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R,16S)-5,9,16-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentanamide
2-[(1,6-dimethyl-4-oxo-1,4-dihydropyridin-3-yl)oxy]-N-(1-methyl-1H-indol-4-yl)acetamide
N-(2,2-dimethyloxan-4-yl)-2-(3-methylbutyl)-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
(4R)-1-[4-(4-methoxyphenyl)piperazin-1-yl]-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R,16S)-5,9,16-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentan-1-one
2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-[2-(5-methoxy-1H-indol-1-yl)ethyl]acetamide
5-methoxy-N-(6-methoxypyridin-3-yl)-4-oxo-4H-pyran-2-carboxamide
2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]-N-(4-methyl-1,3-thiazol-2-yl)acetamide
methyl (2S)-2-[(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)formamido]-4-(methylsulfanyl)butanoate
ethyl 3-(4-hydroxy-2-oxo-1,2-dihydroquinolin-3-yl)-3-[4-(propan-2-yloxy)phenyl]propanoate
2-(7,8-dimethoxy-4-methyl-2-oxo-2H-chromen-3-yl)-N-(2-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}ethyl)acetamide
2-[(7-methoxy-1,2,3,4-tetrahydroacridin-9-yl)sulfanyl]butanedioic acid
(4R)-4-[(1S,2S,5R,7R,10R,11S,14R,15R,16S)-5,16-dihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]-N-(1H-imidazol-2-yl)pentanamide
2-[(4-methyl-2-oxo-2H-chromen-7-yl)oxy]-N-(5-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}pentyl)acetamide
N-(2,2-dimethyloxan-4-yl)-1-(1H-indole-6-carbonyl)piperidine-3-carboxamide
ethyl 3-(4-hydroxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)-3-(2,4,5-trimethoxyphenyl)propanoate
N-[2-(1H-indol-3-yl)ethyl]-3-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
N-{6-[(4-methyl-2-oxo-2H-chromen-7-yl)oxy]pyridin-3-yl}acetamide
5-methoxy-N-[2-(4-methoxyphenyl)ethyl]-4-oxo-4H-pyran-2-carboxamide
(4R)-N-(2,3,4-trifluorophenyl)-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R,16S)-5,9,16-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,7.011,15]heptadecan-14-yl]pentanamide
N-[6-(1H-indol-4-yloxy)pyridin-3-yl]-1-methyl-1H-indole-6-carboxamide hydrochloride
3-{2,3,5,9-tetramethyl-7-oxo-7H-furo[3,2-g]chromen-6-yl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
2-[(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-2H,3H,5H,6H,7H-cyclopenta[c]pyridazin-3-one
2-[(7S)-2,8-dioxo-3,9-diazatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-9-yl]-N-(3,4,5-trimethoxyphenyl)acetamide
N-(1H-imidazol-2-yl)-3-methyl-4-oxo-2-phenyl-4H-chromene-8-carboxamide